SCHEMBL7977591

SCHEMBL7977591

Bc1c(C(=O)OC)[nH]c2ncccc12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 1/20 0.52
KDM4E B2RXH2 5/20 0.44
ALDH1A1 P00352 4/20 0.43
HTT P42858 2/20 0.43
NPSR1 Q6W5P4 2/20 0.43
GAA P10253 1/20 0.43
PADI4 Q9UM07 1/20 0.43
AURKA O14965 1/20 0.41
PARP1 P09874 1/20 0.41
FEN1 P39748 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
HSD17B10 Q99714 2/20 0.39
USP2 O75604 1/20 0.39
TSHR P16473 1/20 0.39
ALOX15 P16050 1/20 0.39
PKM P14618 2/20 0.39
MEN1 O00255 1/20 0.39
TUBB4A P04350 1/20 0.39
TUBB P07437 1/20 0.39
TUBA3C P0DPH7 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7977830 0.83 ALDH1A1 (0.59) MAP2K1KDM4EALDH1A1HTTNPSR1
SCHEMBL7965829 0.83 MAP2K1 (0.54) MAP2K1KDM4EALDH1A1HTTNPSR1
SCHEMBL7975743 0.83 AURKA (0.45) MAP2K1KDM4EALDH1A1NPSR1PADI4
SCHEMBL16496843 0.82 MAP2K1 (0.52) MAP2K1KDM4EALDH1A1HTTNPSR1
SCHEMBL28839540 0.82 MAP2K1 (0.52) MAP2K1KDM4EALDH1A1HTTNPSR1
SCHEMBL1879902 0.82 MAP2K1 (0.52) MAP2K1KDM4EALDH1A1HTTNPSR1
SCHEMBL16497245 0.81 MAP2K1 (0.51) MAP2K1KDM4EALDH1A1HTTNPSR1
SCHEMBL7990805 0.79 MAP2K1 (0.50) MAP2K1KDM4EALDH1A1HTTNPSR1
SCHEMBL24483349 0.78 MAP2K1 (0.49) MAP2K1KDM4EALDH1A1HTTNPSR1
SCHEMBL24483472 0.78 MAP2K1 (0.49) MAP2K1KDM4EALDH1A1HTTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010005528-A2 PYRROLOPYRIDINE CARBOXYLIC ACID DERIVATIVES IRONWOOD PHARMACEUTICALS INCORPORATED (US) 2010-01-14 WO disclosed