SCHEMBL7978780

SCHEMBL7978780

Cc1nc2ccccn2c1-c1ccnc(Nc2nc(C=O)cs2)n1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 11/20 0.62
CDK4 P11802 6/20 0.62
CCNE1 P24864 5/20 0.62
KDM4E B2RXH2 4/20 0.52
ALDH1A1 P00352 4/20 0.52
LMNA P02545 3/20 0.52
MAPT P10636 3/20 0.52
HTT P42858 3/20 0.52
SMN1; SMN2 Q16637 3/20 0.52
GAA P10253 2/20 0.52
NPSR1 Q6W5P4 2/20 0.52
HPGD P15428 2/20 0.52
MEN1 O00255 1/20 0.52
ALOX12 P18054 1/20 0.52
KMT2A Q03164 1/20 0.52
PRKD3 O94806 1/20 0.51
MAP4K4 O95819 1/20 0.51
PIM1 P11309 1/20 0.51
RPS6KB1 P23443 1/20 0.51
FLT4 P35916 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10252038 0.83 CDK2 (0.64) CDK2CDK4CCNE1KDM4EALDH1A1
SCHEMBL701210 0.82 CDK2 (0.60) CDK2CDK4CCNE1KDM4EALDH1A1
SCHEMBL7975583 0.82 CDK2 (0.60) CDK2CDK4CCNE1KDM4EALDH1A1
SCHEMBL7964828 0.80 CDK2 (0.65) CDK2CDK4CCNE1KDM4EALDH1A1
SCHEMBL700855 0.77 HDAC1 (0.64) CDK2CDK4CCNE1PRKD3MAP4K4
SCHEMBL1684673 0.76 CDK2 (0.74) CDK2CDK4CCNE1KDM4EALDH1A1
SCHEMBL7965083 0.76 CDK2 (0.64) CDK2CDK4CCNE1KDM4EALDH1A1
SCHEMBL1684643 0.76 CDK2 (0.86) CDK2CDK4CCNE1KDM4EALDH1A1
SCHEMBL699642 0.75 CDK2 (0.61) CDK2CDK4CCNE1KDM4EALDH1A1
SCHEMBL7964815 0.75 CDK2 (0.63) CDK2CDK4CCNE1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010009155-A2 FUSED HETEROCYCLYC INHIBITOR COMPOUNDS GILEAD COLORADO, INC. (US) 2010-01-21 WO disclosed