SCHEMBL7979834

SCHEMBL7979834

Cc1c(CC(=O)OCc2ccc([N+](=O)[O-])cc2)nc2ccccn12

nearest known ligand 0.50

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.47
PTGS2 P35354 1/20 0.47
MAPT P10636 3/20 0.43
RAB9A P51151 2/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
LMNA P02545 1/20 0.42
ALDH1A1 P00352 1/20 0.41
HTT P42858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7981079 0.76 PTGS1 (0.67) PTGS1PTGS2RAB9ALMNAALDH1A1
SCHEMBL6659912 0.73 ALDH1A1 (0.70) MAPTRAB9AL3MBTL1LMNAALDH1A1
SCHEMBL11688696 0.73 ALDH1A1 (0.70) MAPTRAB9AL3MBTL1LMNAALDH1A1
SCHEMBL7729899 0.72 ALDH1A1 (0.58) MAPTRAB9AL3MBTL1LMNAALDH1A1
SCHEMBL11685951 0.72 MAPT (0.64) MAPTL3MBTL1LMNAALDH1A1
SCHEMBL23783307 0.70 ALDH1A1 (0.64) MAPTRAB9AL3MBTL1ALDH1A1
SCHEMBL28374567 0.69 BCL9 (0.63) MAPTRAB9AL3MBTL1ALDH1A1HTT
SCHEMBL6141237 0.69 ALDH1A1 (0.56) MAPTRAB9AL3MBTL1ALDH1A1HTT
SCHEMBL1555636 0.68 ALDH1A1 (0.59) MAPTRAB9AL3MBTL1ALDH1A1HTT
SCHEMBL20579850 0.68 CYP1A2 (0.75) PTGS1PTGS2MAPTRAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6174877-B1 EXCELLANT BACTERICIDES, ORAL ABSORBABILITY AND STABILITY; IMPROVE THE STABILITY TO RENAL DEHYDROPEPTIDASE I (DHP-I); 2-(2-(N-HETEROCYCLIC-ETHYLTHIO-) DERIVATIVES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-16 US disclosed
EP-0876370-A1 CARBAPENEM COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1998-11-11 EP disclosed
WO-1997025325-A1 CARBAPENEM COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-07-17 WO disclosed