SCHEMBL7979848

SCHEMBL7979848

FC(F)(F)c1ccc(CNc2nc3ccccc3n3cncc23)cc1

nearest known ligand 0.58

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
LCK P06239 16/20 0.58
KDM4E B2RXH2 2/20 0.50
HPGD P15428 2/20 0.50
APP P05067 1/20 0.50
PPARG P37231 1/20 0.50
NR2E3 Q9Y5X4 1/20 0.50
NCOR2 Q9Y618 1/20 0.50
ALDH1A1 P00352 1/20 0.48
THRB P10828 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7980641 0.86 LCK (0.67) LCKKDM4EHPGDALDH1A1THRB
SCHEMBL31500073 0.81 LCK (0.61) LCKKDM4EHPGDAPPALDH1A1
SCHEMBL7987006 0.80 LCK (0.64) LCKKDM4EHPGDALDH1A1
SCHEMBL7986755 0.76 LCK (0.63) LCKKDM4E
SCHEMBL7983552 0.75 LCK (0.67) LCKKDM4EHPGDPPARGNR2E3
SCHEMBL7980569 0.75 KDM4E (0.65) LCKKDM4E
SCHEMBL7969765 0.74 LCK (0.73) LCK
SCHEMBL7980128 0.74 EED (0.61) LCK
SCHEMBL7969596 0.74 LCK (1.00) LCK
SCHEMBL7969734 0.74 LCK (0.58) LCKKDM4EHPGDPPARGNR2E3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235740-B1 AUTOIMMUNE DISEASES; ANTIPROLIFERATION AGENTS BRISTOL-MYERS SQUIBB CO. 2001-05-22 US claimed
WO-1999009845-A1 IMIDAZOQUINOXALINE PROTEIN TYROSINE KINASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 1999-03-04 WO claimed
US-6235740-B1 AUTOIMMUNE DISEASES; ANTIPROLIFERATION AGENTS BRISTOL-MYERS SQUIBB CO. 2001-05-22 US disclosed