SCHEMBL7980285

SCHEMBL7980285

COc1cc2c3ccc(OC)c(OC)c3n(Cc3ccc(Br)cc3)c2cc1OC

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRC P12931 1/20 0.49
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
KDM4E B2RXH2 2/20 0.39
PLA2G2A P14555 1/20 0.38
DRD4 P21917 1/20 0.38
RXFP1 Q9HBX9 2/20 0.37
MAPT P10636 2/20 0.37
PTGS2 P35354 1/20 0.37
PIK3R1 P27986 1/20 0.37
PIK3CA P42336 1/20 0.37
TSHR P16473 2/20 0.36
CYP19A1 P11511 1/20 0.36
NQO2 P16083 1/20 0.36
ALDH1A1 P00352 3/20 0.36
MAPK1 P28482 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
USP2 O75604 1/20 0.36
IDO1 P14902 1/20 0.36
TDO2 P48775 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7970968 0.87 TSHR (0.47) SRCKMT2AKDM4EPLA2G2AMAPT
SCHEMBL7980281 0.84 SRC (0.52) SRCMEN1KMT2AKDM4EDRD4
SCHEMBL7981528 0.84 SRC (0.52) SRCMEN1KMT2AMAPTPIK3R1
SCHEMBL7983968 0.81 SRC (0.56) SRCKMT2AKDM4EMAPTTSHR
SCHEMBL7981648 0.81 SRC (0.53) SRCMEN1KMT2AKDM4ERXFP1
SCHEMBL7983938 0.79 SRC (0.50) SRCKDM4EPLA2G2ARXFP1MAPT
SCHEMBL7971057 0.73 SRC (0.52) SRCKMT2AMAPTPTGS2CYP19A1
SCHEMBL7984408 0.73 SRC (0.51) SRCMEN1KMT2AMAPTALDH1A1
SCHEMBL7984116 0.71 SRC (0.55) SRCPIK3R1PIK3CA
SCHEMBL7980591 0.71 TSHR (0.52) SRCMEN1KMT2AKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6194439-B1 ANTICANCER AGENT PFIZER INC. 2001-02-27 US disclosed
EP-0586608-A1 TRICYCLIC POLYHYDROXYLIC TYROSINE KINASE INHIBITORS PFIZER INC. (US) 1994-03-16 EP disclosed
WO-1992021660-A1 TRICYCLIC POLYHYDROXYLIC TYROSINE KINASE INHIBITORS PFIZER, INC. (US) 1992-12-10 WO disclosed