SCHEMBL7981077

SCHEMBL7981077

CCCC(=O)Oc1nc2ccccn2c1[N+](=O)[O-]

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 2/20 0.58
PTGS2 P35354 2/20 0.58
CYP1A2 P05177 2/20 0.45
LMNA P02545 1/20 0.45
GAA P10253 4/20 0.44
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.44
POLB P06746 1/20 0.44
BCL9 O00512 1/20 0.44
CTNNB1 P35222 1/20 0.44
MAPK1 P28482 1/20 0.41
ALDH1A1 P00352 4/20 0.39
KDM4E B2RXH2 3/20 0.39
DAPK3 O43293 1/20 0.39
JAK2 O60674 1/20 0.39
PRKD3 O94806 1/20 0.39
MAP4K4 O95819 1/20 0.39
ABL1 P00519 1/20 0.39
CSF1R P07333 1/20 0.39
RET P07949 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7979452 0.80 PTGS1 (0.49) PTGS1PTGS2CYP1A2GAAKMT2A
SCHEMBL7981079 0.76 PTGS1 (0.67) PTGS1PTGS2CYP1A2LMNAGAA
SCHEMBL31040146 0.73 PTGS1 (1.00) PTGS1PTGS2CYP1A2LMNAGAA
SCHEMBL10102502 0.72 PTGS1 (0.59) PTGS1PTGS2CYP1A2LMNAGAA
SCHEMBL31040215 0.71 PTGS1 (0.64) PTGS1PTGS2CYP1A2LMNAGAA
SCHEMBL6739461 0.70 PTGS1 (0.61) PTGS1PTGS2CYP1A2LMNAGAA
SCHEMBL7982607 0.69 ADORA2A (0.43) CYP1A2GAAPOLBMAPK1ALDH1A1
SCHEMBL3685087 0.68 PTGS1 (0.61) PTGS1PTGS2CYP1A2LMNAGAA
SCHEMBL29174927 0.68 PTGS1 (0.61) PTGS1PTGS2CYP1A2LMNAGAA
SCHEMBL7980862 0.67 PTGS1 (0.47) PTGS1PTGS2CYP1A2LMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6174877-B1 EXCELLANT BACTERICIDES, ORAL ABSORBABILITY AND STABILITY; IMPROVE THE STABILITY TO RENAL DEHYDROPEPTIDASE I (DHP-I); 2-(2-(N-HETEROCYCLIC-ETHYLTHIO-) DERIVATIVES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-16 US disclosed
EP-0876370-A1 CARBAPENEM COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1998-11-11 EP disclosed
WO-1997025325-A1 CARBAPENEM COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-07-17 WO disclosed