SCHEMBL7979452

SCHEMBL7979452

CCCC(=O)Oc1nc2ccccn2c1N

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 2/20 0.49
PTGS2 P35354 2/20 0.49
DAPK3 O43293 1/20 0.45
JAK2 O60674 1/20 0.45
PRKD3 O94806 1/20 0.45
MAP4K4 O95819 1/20 0.45
ABL1 P00519 1/20 0.45
CSF1R P07333 1/20 0.45
RET P07949 1/20 0.45
MET P08581 1/20 0.45
PDGFRA P16234 1/20 0.45
PRKACA P17612 1/20 0.45
LTK P29376 1/20 0.45
GRK5 P34947 1/20 0.45
KDR P35968 1/20 0.45
MAPK8 P45983 1/20 0.45
MAPK9 P45984 1/20 0.45
CSNK1A1 P48729 1/20 0.45
CDK8 P49336 1/20 0.45
CLK2 P49760 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7981077 0.80 PTGS1 (0.58) PTGS1PTGS2DAPK3JAK2PRKD3
SCHEMBL7979455 0.74 MAPK1 (0.53) PTGS1PTGS2DAPK3JAK2PRKD3
SCHEMBL7982607 0.73 ADORA2A (0.43) MAPK1ALDH1A1KDM4EGAARXFP1
SCHEMBL7982679 0.71 GAA (0.39) DAPK3JAK2PRKD3MAP4K4ABL1
SCHEMBL24611917 0.71 PTGS1 (0.68) PTGS1PTGS2DAPK3JAK2PRKD3
SCHEMBL118200 0.70 PTGS1 (0.65) PTGS1PTGS2DAPK3JAK2PRKD3
SCHEMBL7980862 0.70 PTGS1 (0.47) PTGS1PTGS2MAPK1ALDH1A1KDM4E
SCHEMBL18412790 0.68 PTGS1 (0.73) PTGS1PTGS2DAPK3JAK2PRKD3
SCHEMBL23890512 0.67 PTGS1 (0.50) PTGS1PTGS2DAPK3JAK2PRKD3
SCHEMBL16852188 0.67 ALDH1A1 (0.41) PDGFRAALDH1A1KDM4EGAAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6174877-B1 EXCELLANT BACTERICIDES, ORAL ABSORBABILITY AND STABILITY; IMPROVE THE STABILITY TO RENAL DEHYDROPEPTIDASE I (DHP-I); 2-(2-(N-HETEROCYCLIC-ETHYLTHIO-) DERIVATIVES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-16 US disclosed
EP-0876370-A1 CARBAPENEM COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1998-11-11 EP disclosed
WO-1997025325-A1 CARBAPENEM COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-07-17 WO disclosed