SCHEMBL7981297

SCHEMBL7981297

N=C=O.O=C=Nc1ccc(Cl)c(Cl)c1

nearest known ligand 0.88

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.88
TDP1 Q9NUW8 1/20 0.88
CYP3A4 P08684 3/20 0.44
TRPA1 O75762 1/20 0.44
HTR3E A5X5Y0 2/20 0.42
HTR3B O95264 2/20 0.42
HTR3A P46098 2/20 0.42
HTR3D Q70Z44 2/20 0.42
HTR3C Q8WXA8 2/20 0.42
TSHR P16473 3/20 0.41
KMT2A Q03164 1/20 0.39
ITGB3 P05106 1/20 0.38
ITGAV P06756 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPT P10636 2/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
POLB P06746 1/20 0.37
THRB P10828 1/20 0.37
PMM2 O15305 1/20 0.35
MPI P34949 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL58874 0.94 MAPK1 (1.00) MAPK1TDP1CYP3A4TRPA1HTR3E
SCHEMBL29376406 0.94 MAPK1 (1.00) MAPK1TDP1CYP3A4TRPA1HTR3E
Dimethylamine SCHEMBL11830270 0.86 MAPK1 (0.85) MAPK1TDP1CYP3A4TRPA1HTR3E
SCHEMBL8942897 0.82 TDP1 (0.76) MAPK1TDP1CYP3A4TRPA1HTR3E
SCHEMBL8594415 0.82 TDP1 (0.76) MAPK1TDP1CYP3A4TRPA1HTR3E
O-Xylene SCHEMBL27865799 0.82 MAPK1 (0.76) MAPK1TDP1CYP3A4TRPA1HTR3E
SCHEMBL29709073 0.82 TDP1 (0.70) MAPK1TDP1CYP3A4TRPA1HTR3E
SCHEMBL462305 0.82 TDP1 (0.70) MAPK1TDP1CYP3A4TRPA1HTR3E
SCHEMBL26675676 0.81 MAPK1 (0.63) MAPK1TDP1CYP3A4HTR3EHTR3B
SCHEMBL31347853 0.81 MAPK1 (0.63) MAPK1TDP1CYP3A4HTR3EHTR3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001007431-A2 BENZOTHIOPHENE DERIVATIVES ELI LILLY AND COMPANY (US) 2001-02-01 WO disclosed