SCHEMBL7982419

SCHEMBL7982419

O=C1OC(=O)c2c1ccc1ccc3ccc([N+](=O)[O-])cc3c21

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.58
PTPRC P08575 3/20 0.42
S100A4 P26447 2/20 0.42
BCHE P06276 1/20 0.42
ACHE P22303 1/20 0.42
CES1 P23141 1/20 0.42
CYP1A2 P05177 2/20 0.41
HIF1A Q16665 1/20 0.41
HSD17B10 Q99714 1/20 0.41
CYP3A4 P08684 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
TYMS P04818 2/20 0.39
MAPT P10636 3/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
GABRP O00591 1/20 0.39
GABRD O14764 1/20 0.39
GABRA1 P14867 1/20 0.39
GABRB1 P18505 1/20 0.39
GABRG2 P18507 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4962030 0.90 ALDH1A1 (0.63) ALDH1A1PTPRCS100A4BCHEACHE
SCHEMBL31268201 0.90 ALDH1A1 (0.63) ALDH1A1PTPRCS100A4BCHEACHE
SCHEMBL4960637 0.82 ALDH1A1 (0.61) ALDH1A1PTPRCS100A4BCHEACHE
SCHEMBL7985009 0.78 MAPT (0.56) ALDH1A1TDP1MAPTMEN1KMT2A
SCHEMBL7985135 0.75 TYMS (0.48) ALDH1A1CYP1A2HIF1AHSD17B10CYP3A4
SCHEMBL158311 0.74 ALDH1A1 (1.00) ALDH1A1PTPRCS100A4BCHEACHE
SCHEMBL29661178 0.74 ALDH1A1 (1.00) ALDH1A1PTPRCS100A4BCHEACHE
SCHEMBL9077614 0.74 ALDH1A1 (0.54) ALDH1A1PTPRCS100A4BCHEACHE
SCHEMBL31268251 0.73 ALDH1A1 (0.71) ALDH1A1PTPRCS100A4BCHEACHE
SCHEMBL7971442 0.72 KDM4E (0.44) ALDH1A1HSD17B10TYMSMAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6300340-B1 USEFUL FOR THERAPY OF CANCER AND SOLID TUMORS ADIR ET COMPAGNIE (FR) 2001-10-09 US disclosed
US-6162822-A Bisimide compounds ADIR ET COMPAGNIE (FR) 2000-12-19 US disclosed
EP-0820985-B1 Bis imide derivatives, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 2000-08-30 EP disclosed
EP-0820985-A1 Bis imide derivatives, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1998-01-28 EP disclosed