SCHEMBL7983032

SCHEMBL7983032

C[C@@H](O)[C@H]1C(=O)N2C(C(=O)O)=C(SC(Cc3nccs3)C(O[SiH](C)C)C(C)(C)C)[C@H](C)[C@H]12

nearest known ligand 0.39

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CACNA1C Q13936 1/20 0.37
ESR1 P03372 1/20 0.35
PTGS1 P23219 1/20 0.35
PDE4A P27815 1/20 0.35
FAP Q12884 1/20 0.34
ABCC2 Q92887 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7979861 0.80 CACNA1C (0.42) CACNA1CESR1PTGS1PDE4AFAP
SCHEMBL7983024 0.80 CACNA1C (0.38) CACNA1CESR1PTGS1PDE4AFAP
SCHEMBL7980817 0.79 ESR1 (0.34) CACNA1CESR1PTGS1PDE4AABCC2
SCHEMBL7986586 0.76 CACNA1C (0.42) CACNA1CESR1PTGS1PDE4AFAP
SCHEMBL9026409 0.72 CACNA1C (0.42) CACNA1CESR1PTGS1PDE4AFAP
SCHEMBL9026421 0.72 CACNA1C (0.42) CACNA1CESR1PTGS1PDE4AFAP
SCHEMBL11948525 0.69 CACNA1C (0.35) CACNA1CESR1PTGS1PDE4AFAP
SCHEMBL11956841 0.69 CACNA1C (0.35) CACNA1CESR1PTGS1PDE4AFAP
SCHEMBL21081315 0.68 CACNA1C (0.53) CACNA1CESR1PTGS1PDE4AFAP
SCHEMBL9696922 0.68 CACNA1C (0.50) CACNA1CESR1PTGS1PDE4AFAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6174877-B1 EXCELLANT BACTERICIDES, ORAL ABSORBABILITY AND STABILITY; IMPROVE THE STABILITY TO RENAL DEHYDROPEPTIDASE I (DHP-I); 2-(2-(N-HETEROCYCLIC-ETHYLTHIO-) DERIVATIVES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-16 US disclosed