SCHEMBL7984339

SCHEMBL7984339

NC1(c2ccc(C#Cc3ccc(C(=O)O)cc3)cc2)CC1CCc1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 6/20 0.40
RARB P10826 3/20 0.39
RARG P13631 3/20 0.39
RARA P10276 2/20 0.39
CYP26A1 O43174 1/20 0.39
CYP3A4 P08684 1/20 0.39
CRABP2 P29373 1/20 0.39
FFAR4 Q5NUL3 4/20 0.39
NR4A1 P22736 1/20 0.36
NR4A2 P43354 1/20 0.36
NR4A3 Q92570 1/20 0.36
MMP2 P08253 2/20 0.36
MMP9 P14780 2/20 0.36
MMP12 P39900 2/20 0.36
CHRM2 P08172 1/20 0.36
S1PR1 P21453 1/20 0.36
FPR1 P21462 1/20 0.36
FPR3 P25089 1/20 0.36
GPR183 P32249 1/20 0.36
APLNR P35414 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7984342 0.77 FFAR1 (0.40) FFAR1RARBRARGRARACYP26A1
SCHEMBL5737003 0.71 RARB (0.43) FFAR1RARBRARGRARACYP26A1
SCHEMBL28239851 0.68 SLC1A2 (0.41) FFAR1LMNASLC1A2
SCHEMBL5735140 0.68 NR4A1 (0.49) RARBRARGRARACYP26A1CYP3A4
SCHEMBL5737077 0.68 RARB (0.45) FFAR1RARBRARGRARACYP26A1
SCHEMBL7712760 0.68 RARB (0.45) FFAR1RARBRARGRARACYP26A1
SCHEMBL5737444 0.68 KDM1A (0.47) RARBRARGRARACYP26A1CYP3A4
SCHEMBL402518 0.67 RARB (0.62) FFAR1RARBRARGRARACYP26A1
SCHEMBL6944938 0.66 OPRL1 (0.58) RARBRARGRARACYP26A1CYP3A4
Hydrochloric Acid SCHEMBL2707922 0.66 RARB (0.60) FFAR1RARBRARGRARACYP26A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6303785-B1 SUBSTITUTED N-CYCLOPROPYLTETRAHYDROISOQUINOLINES ALLERGAN SALES, INC. 2001-10-16 US disclosed