SCHEMBL7984582

SCHEMBL7984582

COc1cc2c(nc(N)c3cncn32)c(-c2c(C)cccc2Cl)c1NCCN1CCOCC1

nearest known ligand 0.61

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LCK P06239 12/20 0.61
PDPK1 O15530 1/20 0.48
ALDH1A1 P00352 2/20 0.43
KDM4E B2RXH2 1/20 0.43
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43
ATM Q13315 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
HSD17B10 Q99714 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.41
LYN P07948 2/20 0.40
BTK Q06187 2/20 0.40
POLB P06746 1/20 0.39
SRC P12931 1/20 0.39
MAPK8 P45983 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7980036 0.92 LCK (0.54) LCKPDPK1ALDH1A1KDM4ELMNA
SCHEMBL7982990 0.84 LCK (0.55) LCKPDPK1POLBSRC
SCHEMBL7983111 0.84 LCK (0.58) LCK
SCHEMBL7983651 0.83 LCK (0.59) LCKPDPK1ALDH1A1KDM4ELMNA
SCHEMBL7987022 0.80 LCK (0.52) LCKPDPK1POLBSRC
SCHEMBL4041190 0.80 LCK (0.51) LCKPDPK1ALDH1A1KDM4ELMNA
SCHEMBL7983212 0.79 LCK (0.60) LCKSRC
SCHEMBL7981212 0.78 LCK (0.48) LCKPDPK1POLBSRC
SCHEMBL7983395 0.77 LCK (0.47) LCKPDPK1POLBSRC
SCHEMBL7983616 0.77 LCK (0.51) LCKALDH1A1KDM4ELMNAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235740-B1 AUTOIMMUNE DISEASES; ANTIPROLIFERATION AGENTS BRISTOL-MYERS SQUIBB CO. 2001-05-22 US claimed
WO-1999009845-A1 IMIDAZOQUINOXALINE PROTEIN TYROSINE KINASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 1999-03-04 WO claimed
US-6235740-B1 AUTOIMMUNE DISEASES; ANTIPROLIFERATION AGENTS BRISTOL-MYERS SQUIBB CO. 2001-05-22 US disclosed