SCHEMBL798545

SCHEMBL798545

CCCCCc1nc2c(N3CCNCC3)nc(N)nc2o1

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 18/20 0.45
HRH3 Q9Y5N1 2/20 0.40
KCNH2 Q12809 1/20 0.40
TLR8 Q9NR97 1/20 0.36
TLR7 Q9NYK1 1/20 0.36
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
POLB P06746 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1694230 0.81 HRH4 (0.41) HRH4HRH3KCNH2
SCHEMBL655118 0.77 HRH4 (0.47) HRH4HRH3KCNH2
SCHEMBL655109 0.74 HRH4 (0.45) HRH4HRH3KCNH2TLR8TLR7
SCHEMBL655384 0.72 RAB9A (0.38) TLR8TLR7MEN1ALDH1A1LMNA
SCHEMBL793789 0.71 HRH4 (0.46) HRH4HRH3KCNH2
SCHEMBL605807 0.69 HRH4 (0.47) HRH4HRH3KCNH2TLR8TLR7
SCHEMBL15556511 0.68 HRH4 (0.57) HRH4
SCHEMBL655907 0.67 HRH4 (0.57) HRH4HRH3KCNH2
SCHEMBL602053 0.66 HRH4 (0.44) HRH4HRH3KCNH2ALDH1A1
SCHEMBL605900 0.65 HRH4 (0.48) HRH4HRH3KCNH2MEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2616077-A1 ANTI-CANCER ACTIVITY OF NOVEL BICYCLIC HETEROCYCLES Katholieke Universiteit Leuven, K.U. Leuven R&D (BE) 2013-07-24 EP disclosed
WO-2012035423-A1 ANTI-CANCER ACTIVITY OF NOVEL BICYCLIC HETEROCYCLES KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2012-03-22 WO disclosed