SCHEMBL7986168

SCHEMBL7986168

O=Cc1cnc2cccc(Cl)n12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1B Q9Y463 2/20 0.41
CHEK1 O14757 1/20 0.41
LTK P29376 1/20 0.41
GRK5 P34947 1/20 0.41
CSNK1A1 P48729 1/20 0.41
LIMK1 P53667 1/20 0.41
TYRO3 Q06418 1/20 0.41
LRRK2 Q5S007 1/20 0.41
CLK4 Q9HAZ1 1/20 0.41
LMNA P02545 2/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
POLB P06746 1/20 0.38
ALDH1A1 P00352 2/20 0.36
DYRK3 O43781 1/20 0.35
CCNT1 O60563 1/20 0.35
CDK9 P50750 1/20 0.35
CDK5 Q00535 1/20 0.35
DYRK1A Q13627 1/20 0.35
CDK5R1 Q15078 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11880227 0.79 ALDH1A1 (0.33) DYRK1BCHEK1LTKGRK5CSNK1A1
SCHEMBL16033029 0.79 HTT (0.39) KMT2APOLBALDH1A1ATMGAA
SCHEMBL30431689 0.75 DYRK1A (0.33) DYRK1BPOLBALDH1A1DYRK1ADYRK2
SCHEMBL16506228 0.72 DYRK1B (0.44) DYRK1BCHEK1LTKGRK5CSNK1A1
SCHEMBL30063374 0.71 TRIM24 (0.37) KMT2APOLBALDH1A1ATMHTT
SCHEMBL2549330 0.67 NPSR1 (0.50) POLBALDH1A1DYRK1AATMGAA
SCHEMBL14639038 0.66 MKNK1 (0.49) DYRK1BALDH1A1DYRK3CCNT1CDK9
SCHEMBL15549142 0.65 KMT2A (0.38) LMNAMEN1KMT2AALDH1A1ATM
SCHEMBL5100079 0.64 POLB (0.47) MEN1KMT2APOLBALDH1A1GAA
SCHEMBL1163131 0.64 DYRK1A (0.54) DYRK1BALDH1A1DYRK3CCNT1CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed
US-6235731-B1 REDUCING BLOOD LIPIDS, SUGARS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-22 US disclosed
EP-0915888-A1 FUSED IMIDAZOPYRIDINE DERIVATIVES AS ANTIHYPERLIPIDEMIC AGENTS Takeda Chemical Industries, Ltd. (JP) 1999-05-19 EP disclosed
WO-1998025926-A1 IMIDAZOPYRIDINE DERIVATIVES AND THEIR PRODUCTION TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-06-18 WO disclosed
WO-1997040051-A1 FUSED IMIDAZOPYRIDINE DERIVATIVES AS ANTIHYPERLIPIDEMIC AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-10-30 WO disclosed