SCHEMBL7986602

SCHEMBL7986602

CC(C)[C@H]1COC(=O)N1C(=O)Cc1ccc2c(c1)OCO2

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.47
CYP3A4 P08684 3/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2C19 P33261 1/20 0.47
IL6ST P40189 2/20 0.46
KDM4E B2RXH2 1/20 0.45
HTT P42858 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.43
TAAR1 Q96RJ0 2/20 0.42
SLC6A2 P23975 2/20 0.42
SLC6A3 Q01959 2/20 0.42
SLC6A4 P31645 1/20 0.42
CMA1 P23946 1/20 0.42
GAA P10253 1/20 0.42
HSD17B10 Q99714 1/20 0.42
HPGD P15428 1/20 0.41
SIGMAR1 Q99720 2/20 0.41
LMNA P02545 1/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8225610 0.81 IL6ST (0.52) ALDH1A1IL6STHTTSMN1; SMN2HPGD
SCHEMBL19183081 0.81 IL6ST (0.52) ALDH1A1IL6STHTTSMN1; SMN2
SCHEMBL4775861 0.81 IL6ST (0.52) ALDH1A1IL6STHTTSMN1; SMN2
SCHEMBL4767686 0.81 IL6ST (0.52) ALDH1A1IL6STHTTSMN1; SMN2
SCHEMBL4767695 0.81 IL6ST (0.52) ALDH1A1CYP2C19IL6STHPGDTSHR
SCHEMBL4770816 0.81 IL6ST (0.52) ALDH1A1CYP2C19IL6STHPGDTSHR
SCHEMBL5108652 0.81 HTT (0.51) ALDH1A1CYP2C19IL6STKDM4EHTT
SCHEMBL5108649 0.81 HTT (0.51) ALDH1A1CYP2C19IL6STKDM4EHTT
SCHEMBL14032439 0.81 HTT (0.51) ALDH1A1CYP2C19IL6STKDM4EHTT
SCHEMBL9970272 0.80 IL6ST (0.66) ALDH1A1IL6STKDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6207686-B1 FOR THERAPY OF HYPERTENSION FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-03-27 US disclosed
EP-0792265-A1 ENDOTHELIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-09-03 EP disclosed
WO-1996015109-A1 ENDOTHELIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-05-23 WO disclosed