SCHEMBL7986774

SCHEMBL7986774

CCOc1ccc([C@@H](CC(=O)O)N(C(C)=O)N2C(=O)N[C@](C)(c3ccc(C(=N)N)cc3)C2=O)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 7/20 0.46
ITGA2B P08514 7/20 0.46
PRSS1 P07477 2/20 0.40
PRSS2 P07478 2/20 0.40
PRSS3 P35030 2/20 0.40
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
CRHBP P24387 1/20 0.38
CRHR2 Q13324 1/20 0.38
F10 P00742 3/20 0.36
F7 P08709 2/20 0.36
F3 P13726 2/20 0.36
ALDH1A1 P00352 2/20 0.34
POLB P06746 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
TP53 P04637 1/20 0.34
TSHR P16473 1/20 0.34
PARP10 Q53GL7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7981888 0.90 ITGB3 (0.50) ITGB3ITGA2BMEN1KMT2ACYP2C9
SCHEMBL7985139 0.89 ITGB3 (0.49) ITGB3ITGA2BMEN1KMT2AF7
Hydrochloric Acid SCHEMBL7969557 0.88 ITGB3 (0.56) ITGB3ITGA2BMEN1KMT2AF10
Hydrochloric Acid SCHEMBL8489120 0.88 ITGB3 (0.56) ITGB3ITGA2BMEN1KMT2AF10
Hydrochloric Acid SCHEMBL7986512 0.88 ITGB3 (0.56) ITGB3ITGA2BMEN1KMT2AF10
Hydrochloric Acid SCHEMBL8488362 0.88 ITGB3 (0.56) ITGB3ITGA2BMEN1KMT2AF10
SCHEMBL8489046 0.87 ITGB3 (0.52) ITGB3ITGA2BMEN1KMT2AALDH1A1
SCHEMBL7451749 0.85 MEN1 (0.39) ITGB3ITGA2BMEN1KMT2ACRHBP
SCHEMBL7969575 0.84 ITGB3 (0.45) ITGB3ITGA2BPRSS1PRSS2PRSS3
SCHEMBL8492974 0.84 ITGB3 (0.45) ITGB3ITGA2BPRSS1PRSS2PRSS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6191282-B1 DERIVATIVES OF 5-MEMBERED NITROGEN CONTAINING HETEROCYCLIC RING IS USED AS ANTICARCINOGENIC AGENT AND ANTICOAGULANT HOECHST MARION ROUSSEL (DE) 2001-02-20 US disclosed
US-5981492-A ADMINISTERED TO THE PATIENT TO INHIBIT THROMBOCYTE AGGREGATION, THE METASTASIZATION OF CARCINOMA CELLS, THE BINDING OF OSTEOCLASTS TO THE BONE SURFACE, OR FOR THE TREATMENT OF THROMBOSES HOECHST AKTIENGESELLSCHAFT (DE) 1999-11-09 US disclosed