SCHEMBL7986855

SCHEMBL7986855

COC(=O)Cc1nnc2ccccn12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.56
ALDH1A1 P00352 3/20 0.56
RAB9A P51151 6/20 0.47
NPC1 O15118 4/20 0.47
SMN1; SMN2 Q16637 3/20 0.46
HPGD P15428 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
DAPK3 O43293 1/20 0.43
JAK2 O60674 1/20 0.43
PRKD3 O94806 1/20 0.43
MAP4K4 O95819 1/20 0.43
ABL1 P00519 1/20 0.43
CSF1R P07333 1/20 0.43
RET P07949 1/20 0.43
MET P08581 1/20 0.43
PDGFRA P16234 1/20 0.43
PRKACA P17612 1/20 0.43
LTK P29376 1/20 0.43
GRK5 P34947 1/20 0.43
KDR P35968 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21577704 0.85 ALDH1A1 (0.53) KDM4EALDH1A1RAB9ANPC1SMN1; SMN2
SCHEMBL7980785 0.81 KDM4E (0.62) KDM4EALDH1A1RAB9ANPC1SMN1; SMN2
SCHEMBL21577705 0.80 KDM4E (0.61) KDM4EALDH1A1RAB9ANPC1SMN1; SMN2
SCHEMBL5373208 0.77 KDM4E (0.71) KDM4EALDH1A1RAB9ANPC1SMN1; SMN2
SCHEMBL5354841 0.76 KDM4E (0.56) KDM4EALDH1A1RAB9ANPC1SMN1; SMN2
SCHEMBL20434857 0.75 GGPS1 (0.50) KDM4EALDH1A1RAB9ANPC1SMN1; SMN2
SCHEMBL7981341 0.75 ALDH1A1 (0.46) KDM4EALDH1A1RAB9ANPC1SMN1; SMN2
SCHEMBL13341900 0.74 ALDH1A1 (0.61) KDM4EALDH1A1SMN1; SMN2HPGDCYP2C9
SCHEMBL8350565 0.73 KDM4E (0.71) KDM4EALDH1A1RAB9ANPC1SMN1; SMN2
SCHEMBL12797503 0.72 KDM4E (0.70) KDM4EALDH1A1RAB9ANPC1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6174877-B1 EXCELLANT BACTERICIDES, ORAL ABSORBABILITY AND STABILITY; IMPROVE THE STABILITY TO RENAL DEHYDROPEPTIDASE I (DHP-I); 2-(2-(N-HETEROCYCLIC-ETHYLTHIO-) DERIVATIVES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-16 US disclosed
EP-0876370-A1 CARBAPENEM COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1998-11-11 EP disclosed
WO-1997025325-A1 CARBAPENEM COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-07-17 WO disclosed