SCHEMBL7987389

SCHEMBL7987389

O=C(NNC(=O)c1cccnc1)Nc1cccc2c1C(=O)c1c-2n[nH]c1-c1ccc(N2CCNCC2)cc1

nearest known ligand 0.53

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 15/20 0.53
CCND1 P24385 15/20 0.53
CDK2 P24941 14/20 0.53
CCNE2 O96020 13/20 0.53
CCNE1 P24864 13/20 0.53
ALDH1A1 P00352 2/20 0.44
KDM4E B2RXH2 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C19 P33261 1/20 0.42
MAPT P10636 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8003499 0.92 CDK4 (0.54) CDK4CCND1CDK2CCNE2CCNE1
SCHEMBL7987302 0.92 CDK4 (0.55) CDK4CCND1CDK2CCNE2CCNE1
SCHEMBL7987393 0.87 CDK2 (0.49) CDK4CCND1CDK2CCNE2CCNE1
SCHEMBL8003502 0.86 CCNE2 (0.60) CDK4CCND1CDK2CCNE2CCNE1
SCHEMBL7998047 0.85 CCNE2 (0.65) CDK4CCND1CDK2CCNE2CCNE1
SCHEMBL6349463 0.84 CDK4 (0.52) CDK4CCND1CDK2CCNE2CCNE1
SCHEMBL5524473 0.83 CCNE2 (0.74) CDK4CCND1CDK2CCNE2CCNE1
SCHEMBL8003511 0.83 CDK4 (0.56) CDK4CCND1CDK2CCNE2CCNE1
SCHEMBL4028350 0.83 CDK4 (0.59) CDK4CCND1CDK2CCNE2CCNE1
SCHEMBL4027332 0.81 CCNE2 (0.59) CDK4CCND1CDK2CCNE2CCNE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6291504-B1 POTENT INHIBITORS OF THE CLASS OF ENZYMES KNOWN AS CYCLIN DEPENDENT KINASES DUPONT PHARMACEUTICALS COMPANY 2001-09-18 US claimed
US-6291504-B1 POTENT INHIBITORS OF THE CLASS OF ENZYMES KNOWN AS CYCLIN DEPENDENT KINASES DUPONT PHARMACEUTICALS COMPANY 2001-09-18 US disclosed