SCHEMBL8003511

SCHEMBL8003511

CN1CCN(c2ccc(-c3[nH]nc4c3C(=O)c3c(NC(=O)NNC(=O)c5ccncc5)cccc3-4)cc2)CC1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 19/20 0.56
CCND1 P24385 19/20 0.56
CDK2 P24941 14/20 0.56
CCNE2 O96020 13/20 0.56
CCNE1 P24864 13/20 0.56
CCNB2 O95067 1/20 0.50
ABL1 P00519 1/20 0.50
CDK1 P06493 1/20 0.50
CCNB1 P14635 1/20 0.50
CCNA2 P20248 1/20 0.50
CCNA1 P78396 1/20 0.50
CCNB3 Q8WWL7 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8003514 0.94 CCNE2 (0.62) CDK4CCND1CDK2CCNE2CCNE1
SCHEMBL8003499 0.92 CDK4 (0.54) CDK4CCND1CDK2CCNE2CCNE1
SCHEMBL7987302 0.91 CDK4 (0.55) CDK4CCND1CDK2CCNE2CCNE1
SCHEMBL8003502 0.85 CCNE2 (0.60) CDK4CCND1CDK2CCNE2CCNE1
SCHEMBL7664909 0.84 CDK4 (0.69) CDK4CCND1CDK2CCNE2CCNE1
SCHEMBL5514242 0.84 CCNE2 (0.78) CDK4CCND1CDK2CCNE2CCNE1
SCHEMBL7662345 0.84 CDK4 (0.63) CDK4CCND1CDK2CCNE2CCNE1
SCHEMBL7987389 0.83 CDK4 (0.53) CDK4CCND1CDK2CCNE2CCNE1
SCHEMBL4025333 0.82 CDK4 (0.69) CDK4CCND1CDK2CCNE2CCNE1
SCHEMBL6346628 0.81 CDK4 (0.52) CDK4CCND1CDK2CCNE2CCNE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6291504-B1 POTENT INHIBITORS OF THE CLASS OF ENZYMES KNOWN AS CYCLIN DEPENDENT KINASES DUPONT PHARMACEUTICALS COMPANY 2001-09-18 US claimed
US-6291504-B1 POTENT INHIBITORS OF THE CLASS OF ENZYMES KNOWN AS CYCLIN DEPENDENT KINASES DUPONT PHARMACEUTICALS COMPANY 2001-09-18 US disclosed