SCHEMBL7987902

SCHEMBL7987902

COc1ccc2c(c1)c(-c1cncc(-c3cccc(Cl)c3)c1)cn2CCN1CCOCC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 3/20 0.53
FLT1 P17948 2/20 0.53
FLT4 P35916 2/20 0.53
CNR2 P34972 5/20 0.47
MKNK2 Q9HBH9 1/20 0.43
PDE4B Q07343 1/20 0.43
CYP1A2 P05177 2/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2D6 P10635 2/20 0.43
LMNA P02545 1/20 0.43
TP53 P04637 1/20 0.43
ALOX15 P16050 1/20 0.43
HIF1A Q16665 1/20 0.43
HSD17B10 Q99714 1/20 0.43
HTR6 P50406 1/20 0.42
NFATC1 O95644 1/20 0.41
GSK3B P49841 1/20 0.41
DYRK1A Q13627 1/20 0.41
CNR1 P21554 3/20 0.41
PDE2A O00408 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7976794 0.93 KDR (0.53) KDRFLT1FLT4CNR2MKNK2
SCHEMBL7990446 0.93 KDR (0.56) KDRFLT1FLT4CNR2MKNK2
SCHEMBL7548695 0.92 KDR (0.52) KDRFLT1FLT4CNR2HSD17B10
SCHEMBL7990472 0.90 KDR (0.53) KDRFLT1FLT4CNR2MKNK2
SCHEMBL7991015 0.90 KDR (0.59) KDRFLT1FLT4CNR2MKNK2
SCHEMBL7976802 0.90 KDR (0.59) KDRFLT1FLT4CNR2LMNA
SCHEMBL7990519 0.88 KDR (0.53) KDRFLT1FLT4CNR2MKNK2
SCHEMBL7550594 0.88 KDR (0.56) KDRFLT1FLT4CNR2MKNK2
SCHEMBL7986681 0.88 KDR (0.53) KDRFLT1FLT4CNR2MKNK2
SCHEMBL7549728 0.87 KDR (0.54) KDRFLT1FLT4GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed