SCHEMBL7991015

SCHEMBL7991015

COc1ccc2c(c1)c(-c1cncc(-c3ccccc3)c1)cn2CCN1CCOCC1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 5/20 0.59
FLT1 P17948 3/20 0.59
FLT4 P35916 3/20 0.59
CNR2 P34972 3/20 0.51
HTR6 P50406 1/20 0.49
MKNK2 Q9HBH9 1/20 0.48
GSK3B P49841 2/20 0.45
NFATC1 O95644 1/20 0.45
DYRK1A Q13627 1/20 0.45
PTPN1 P18031 1/20 0.44
CNR1 P21554 1/20 0.44
LMNA P02545 1/20 0.44
TP53 P04637 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
ALOX15 P16050 1/20 0.44
HIF1A Q16665 1/20 0.44
HSD17B10 Q99714 1/20 0.44
CYP11B1 P15538 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7550594 0.94 KDR (0.56) KDRFLT1FLT4CNR2HTR6
SCHEMBL7990446 0.93 KDR (0.56) KDRFLT1FLT4CNR2HTR6
SCHEMBL7550504 0.91 KDR (0.59) KDRFLT1FLT4CNR2HTR6
SCHEMBL7990472 0.91 KDR (0.53) KDRFLT1FLT4CNR2HTR6
SCHEMBL7987902 0.90 KDR (0.53) KDRFLT1FLT4CNR2HTR6
SCHEMBL7990662 0.89 KDR (0.68) KDRFLT1FLT4CNR2MKNK2
SCHEMBL7990934 0.88 KDR (0.66) KDRFLT1FLT4MKNK2GSK3B
SCHEMBL7987864 0.87 KDR (0.74) KDRFLT1FLT4CNR2HTR6
SCHEMBL7990519 0.87 KDR (0.53) KDRFLT1FLT4CNR2MKNK2
SCHEMBL7976794 0.86 KDR (0.53) KDRFLT1FLT4CNR2MKNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed