SCHEMBL7987912

SCHEMBL7987912

CCCN(CCC)C(=O)c1ccc2c(c1)C(=C(Nc1ccc(Cl)cc1)c1ccccc1)C(=O)N2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 1/20 0.40
PAK4 O96013 3/20 0.40
KDR P35968 3/20 0.38
TP53 P04637 1/20 0.38
LRRK2 Q5S007 1/20 0.38
EGFR P00533 1/20 0.38
INSR P06213 1/20 0.38
IGF1R P08069 1/20 0.38
PDGFRB P09619 1/20 0.38
KIT P10721 1/20 0.38
FGFR1 P11362 1/20 0.38
SRC P12931 1/20 0.38
PDGFRA P16234 1/20 0.38
FLT1 P17948 1/20 0.38
EPHA2 P29317 1/20 0.38
FLT4 P35916 1/20 0.38
FLT3 P36888 1/20 0.38
RPS6KA3 P51812 1/20 0.38
EPHB4 P54760 1/20 0.38
KCNH2 Q12809 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6980882 1.00 TLR8 (0.40) TLR8PAK4KDRTP53LRRK2
SCHEMBL6978234 0.93 TP53 (0.41) TLR8PAK4TP53LIMK1LIMK2
SCHEMBL6978230 0.93 TP53 (0.41) TLR8PAK4TP53LIMK1LIMK2
SCHEMBL7226471 0.89 LRRK2 (0.42) TLR8PAK4KDRLRRK2EGFR
SCHEMBL7226468 0.89 LRRK2 (0.42) TLR8PAK4KDRLRRK2EGFR
SCHEMBL6975580 0.88 HDAC1 (0.43) TP53LIMK1LIMK2HDAC1HDAC6
SCHEMBL6975585 0.88 HDAC1 (0.43) TP53LIMK1LIMK2HDAC1HDAC6
SCHEMBL6985372 0.88 HDAC1 (0.42) LIMK1LIMK2NAMPTHDAC1HDAC6
SCHEMBL6985368 0.88 HDAC1 (0.42) LIMK1LIMK2NAMPTHDAC1HDAC6
SCHEMBL7985455 0.88 JAK3 (0.44) PAK4KDRLRRK2FLT3RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6169106-B1 ANTITUMOUR AGENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 2001-01-02 US disclosed