SCHEMBL6985372

SCHEMBL6985372

CCCN(CCC)C(=O)c1ccc2c(c1)C(=C(Nc1ccc(CN(C)Cc3ccccc3)cc1)c1ccccc1)C(=O)N2

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
ALDH1A1 P00352 1/20 0.42
ACHE P22303 5/20 0.41
BCHE P06276 3/20 0.41
LIMK1 P53667 2/20 0.39
RORC P51449 2/20 0.38
LTA4H P09960 1/20 0.38
NAMPT P43490 1/20 0.38
LIMK2 P53671 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6985368 1.00 HDAC1 (0.42) HDAC1HDAC6ALDH1A1ACHEBCHE
SCHEMBL6975585 0.94 HDAC1 (0.43) HDAC1HDAC6ALDH1A1LIMK1RORC
SCHEMBL6975580 0.94 HDAC1 (0.43) HDAC1HDAC6ALDH1A1LIMK1RORC
SCHEMBL6983164 0.93 ACHE (0.45) HDAC1HDAC6ACHEBCHERORC
SCHEMBL6983168 0.93 ACHE (0.45) HDAC1HDAC6ACHEBCHERORC
SCHEMBL7233846 0.92 ALDH1A1 (0.45) HDAC1HDAC6ALDH1A1ACHEBCHE
SCHEMBL7233848 0.92 ALDH1A1 (0.45) HDAC1HDAC6ALDH1A1ACHEBCHE
SCHEMBL6979863 0.90 ACHE (0.44) HDAC1ACHEBCHERORCLTA4H
SCHEMBL6979865 0.90 ACHE (0.44) HDAC1ACHEBCHERORCLTA4H
SCHEMBL6978234 0.90 TP53 (0.41) HDAC1HDAC6ALDH1A1LIMK1NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1071665-B1 SUBSTITUTED INDOLINONES HAVING AN INHIBITING EFFECT ON KINASES AND CYCLINE/CDK COMPLEXES BOEHRINGER INGELHEIM PHARMA (DE) 2003-10-01 EP disclosed
EP-1071665-A1 SUBSTITUTED INDOLINONES HAVING AN INHIBITING EFFECT ON KINASES AND CYCLINE/CDK COMPLEXES Boehringer Ingelheim Pharma KG (DE) 2001-01-31 EP disclosed
WO-1999052869-A1 SUBSTITUTED INDOLINONES HAVING AN INHIBITING EFFECT ON KINASES AND CYCLINE/CDK COMPLEXES BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-10-21 WO disclosed