SCHEMBL7988067

SCHEMBL7988067

COCn1cc(C2=C(c3cn(C)c4cc([N+](=O)[O-])ccc34)C(=O)NC2=O)c2ccc(N3CCCC3)cc21

nearest known ligand 0.59

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 5/20 0.39
QPCT Q16769 2/20 0.39
PRKCA P17252 3/20 0.39
KDR P35968 1/20 0.38
FLT3 P36888 1/20 0.38
CCNE2 O96020 1/20 0.38
CDK4 P11802 1/20 0.38
CCND1 P24385 1/20 0.38
CCNE1 P24864 1/20 0.38
CDK2 P24941 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7988030 0.91 CDK4 (0.45) GSK3BCCNE2CDK4CCND1CCNE1
SCHEMBL6948330 0.85 CCNE2 (0.54) GSK3BQPCTCCNE2CDK4CCND1
SCHEMBL7976559 0.83 GSK3B (0.53) GSK3BPRKCACCNE2CDK4CCND1
SCHEMBL7599053 0.82 CCNE2 (0.51) PRKCACCNE2CDK4CCND1CCNE1
SCHEMBL668748 0.80 CCNE2 (0.57) CCNE2CDK4CCND1CCNE1CDK2
SCHEMBL7988158 0.78 GSK3B (0.51) GSK3BPRKCAKDRCCNE2CDK4
SCHEMBL7990678 0.77 GSK3B (0.59) GSK3BPRKCAKDRCCNE2CDK4
SCHEMBL7059442 0.76 GSK3B (0.57) GSK3BPRKCACCNE2CDK4CCND1
SCHEMBL7976776 0.76 CDK4 (0.67) GSK3BPRKCACCNE2CDK4CCND1
SCHEMBL7508119 0.76 CCNE2 (0.56) CCNE2CDK4CCND1CCNE1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6281356-B1 ANTICANRCER AGENTS HOFFMANN-LA ROCHE INC. 2001-08-28 US claimed
US-6281356-B1 ANTICANRCER AGENTS HOFFMANN-LA ROCHE INC. 2001-08-28 US disclosed