SCHEMBL7989760

SCHEMBL7989760

O=C(O)c1ccc(C(O)C(C(=O)O)c2ccc3c(c2)OCO3)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.59
MAPK1 P28482 2/20 0.59
SRD5A2 P31213 1/20 0.57
MAPK9 P45984 1/20 0.54
CYP1A2 P05177 2/20 0.46
CYP2C9 P11712 2/20 0.46
CYP2C19 P33261 2/20 0.46
PTGS1 P23219 1/20 0.46
PTGS2 P35354 1/20 0.46
NPC1 O15118 4/20 0.45
RAB9A P51151 3/20 0.45
PAX8 Q06710 2/20 0.45
L3MBTL1 Q9Y468 2/20 0.45
LMNA P02545 1/20 0.45
GAA P10253 1/20 0.45
MAPT P10636 1/20 0.45
CTNNB1 P35222 1/20 0.43
WNT3A P56704 1/20 0.43
KMT2A Q03164 2/20 0.43
CA12 O43570 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7990464 0.90 MAPK9 (0.54) ALDH1A1MAPK1SRD5A2MAPK9CYP1A2
SCHEMBL7987319 0.88 MAPK1 (0.50) ALDH1A1MAPK1MAPK9CYP1A2CYP2C9
SCHEMBL7987077 0.85 NPC1 (0.55) ALDH1A1MAPK1MAPK9CYP1A2CYP2C9
SCHEMBL7976622 0.84 MAPK9 (0.47) ALDH1A1MAPK1MAPK9CYP1A2CYP2C9
SCHEMBL8035766 0.77 PTGS1 (0.59) ALDH1A1MAPK1MAPK9CYP1A2CYP2C9
SCHEMBL29785806 0.77 MAPK9 (0.56) ALDH1A1MAPK1SRD5A2MAPK9CYP1A2
SCHEMBL1154990 0.77 MAPK9 (0.56) ALDH1A1MAPK1SRD5A2MAPK9CYP1A2
SCHEMBL4510613 0.77 MAPK9 (0.56) ALDH1A1MAPK1SRD5A2MAPK9CYP1A2
SCHEMBL22722996 0.77 MAPK9 (0.56) ALDH1A1MAPK1SRD5A2MAPK9CYP1A2
SCHEMBL7993658 0.77 KMT2A (0.49) ALDH1A1MAPK1L3MBTL1LMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265473-B1 STABILIZER; HEAT AND OXIDATION RESISTANCE; PHOTOSTABILITY CIBA SPECIALTY CHEMICALS CORP. 2001-07-24 US disclosed
US-6207686-B1 FOR THERAPY OF HYPERTENSION FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-03-27 US disclosed
WO-1996015109-A1 ENDOTHELIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-05-23 WO disclosed