SCHEMBL7989812

SCHEMBL7989812

COc1cccc(N2CCN(CCCCN3CSCC3=O)CC2)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.67
HTR1A P08908 7/20 0.61
DRD2 P14416 4/20 0.60
DRD1 P21728 1/20 0.60
DRD3 P35462 1/20 0.60
HTR2A P28223 2/20 0.56
HTR7 P34969 2/20 0.56
ADRA2A P08913 1/20 0.56
ADRA2C P18825 1/20 0.56
DRD4 P21917 1/20 0.56
HRH2 P25021 1/20 0.56
HTR1B P28222 1/20 0.56
ADRA1A P35348 1/20 0.56
HRH1 P35367 1/20 0.56
ADRA1B P35368 1/20 0.56
HTR2B P41595 1/20 0.56
SIGMAR1 Q99720 1/20 0.56
HTR6 P50406 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7989785 0.99 KCNH2 (0.66) KCNH2HTR1ADRD2DRD1DRD3
SCHEMBL7996696 0.86 KCNH2 (0.66) KCNH2
Hydrochloric Acid SCHEMBL7979104 0.85 KCNH2 (0.64) KCNH2
SCHEMBL7997136 0.85 KCNH2 (0.67) KCNH2
Hydrochloric Acid SCHEMBL7990518 0.84 KCNH2 (0.66) KCNH2
SCHEMBL4525293 0.82 KCNH2 (1.00) KCNH2HTR1ADRD2DRD1DRD3
SCHEMBL7991242 0.81 HTR7 (0.65) DRD2DRD1DRD3HTR7SIGMAR1
Hydrochloric Acid SCHEMBL7993795 0.80 HTR7 (0.62) DRD2DRD1DRD3HTR7SIGMAR1
Hydrochloric Acid SCHEMBL7993796 0.80 HTR7 (0.62) DRD2DRD1DRD3HTR7SIGMAR1
SCHEMBL7990544 0.79 HTR7 (0.66) HTR1ADRD2DRD3HTR7DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6284775-B1 PSYCHOLOGICAL DISORDERS AVENTIS PHARMACEUTICALS INC. 2001-09-04 US disclosed
US-5371087-A Antipsychotic, analgesics, anticonvulsant and anxiolytic agent HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-12-06 US disclosed
US-5229388-A 3-[4-(1-substituted-4-piperazinyl)butyl]-4-thiazolidinone and related compounds HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-07-20 US disclosed
EP-0316723-B1 3-[4(1-Substituted-4-piperazinyl)butyl]-4-thiazolidinones a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-09-30 EP disclosed
US-5136037-A 3-(4-substituted-4-piperazinyl)butyl-4-thiazolidinone and related compounds HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1992-08-04 US disclosed
US-5037984-A Anticonvulsants; anxiolytic agents HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1991-08-06 US disclosed
US-4933453-A ANTIPSYCHOTIC, ANALGESIC, ANTICONVULSANT, AND ANXIOLYTIC AGENTS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1990-06-12 US disclosed
EP-0316723-A1 3-[4(1-Substituted-4-piperazinyl)butyl]-4-thiazolidinones a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-05-24 EP disclosed