SCHEMBL7990118

SCHEMBL7990118

COc1cccc2c(-c3cncc(-c4cccc(Cl)c4)c3)cn(C(C)CN(C)C)c12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 2/20 0.39
FLT1 P17948 1/20 0.39
FLT4 P35916 1/20 0.39
PDE4B Q07343 4/20 0.36
FYN P06241 1/20 0.36
PDE4D Q08499 1/20 0.35
HCRTR1 O43613 1/20 0.35
HCRTR2 O43614 1/20 0.35
MAPK10 P53779 3/20 0.34
GRIN2B Q13224 1/20 0.34
KMT2A Q03164 1/20 0.34
HTR6 P50406 1/20 0.34
RIPK2 O43353 1/20 0.34
LYN P07948 1/20 0.34
TAAR1 Q96RJ0 1/20 0.33
DPP4 P27487 1/20 0.33
ALPL P05186 1/20 0.33
MAPK9 P45984 1/20 0.33
MAPK14 Q16539 1/20 0.33
CNR2 P34972 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7549333 0.90 KDR (0.43) KDRFLT1FLT4HCRTR1HCRTR2
SCHEMBL7546645 0.89 FLT1 (0.40) KDRFLT1FLT4FYNHTR6
SCHEMBL7546769 0.87 KDR (0.51) KDRFLT1FLT4PDE4BFYN
SCHEMBL7549222 0.86 KDR (0.40) KDRFLT1FLT4HTR6ALPL
SCHEMBL7549609 0.85 KDR (0.49) KDRFLT1FLT4GRIN2BKMT2A
SCHEMBL7990227 0.84 PDE4B (0.45) KDRFLT1FLT4PDE4BPDE4D
SCHEMBL7990501 0.84 KDR (0.58) KDRFLT1FLT4ALPLCNR2
SCHEMBL7994139 0.83 KDR (0.41) KDRFLT1FLT4PDE4BPDE4D
SCHEMBL7988607 0.83 KDR (0.43) KDRFLT1FLT4GRIN2BTAAR1
SCHEMBL7994193 0.81 KDR (0.49) KDRFLT1FLT4PDE4BFYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed