SCHEMBL7990501

SCHEMBL7990501

COc1cccc2c(-c3cncc(-c4ccsc4)c3)cn(C(C)CN(C)C)c12

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 8/20 0.58
FLT1 P17948 4/20 0.58
FLT4 P35916 4/20 0.58
CYP2A6 P11509 3/20 0.40
PDGFRB P09619 2/20 0.36
PDGFRA P16234 2/20 0.36
ALPL P05186 1/20 0.35
ADRA2A P08913 3/20 0.34
ADRA2B P18089 3/20 0.34
ADRA2C P18825 3/20 0.34
TUBB4A P04350 2/20 0.33
TUBB P07437 2/20 0.33
TUBA3C P0DPH7 2/20 0.33
TUBA1B P68363 2/20 0.33
TUBA4A P68366 2/20 0.33
TUBB4B P68371 2/20 0.33
TUBB3 Q13509 2/20 0.33
TUBB2A Q13885 2/20 0.33
TUBB8 Q3ZCM7 2/20 0.33
TUBA3E Q6PEY2 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7990474 0.87 KDR (0.71) KDRFLT1FLT4CYP2A6PDGFRB
SCHEMBL7549333 0.87 KDR (0.43) KDRFLT1FLT4CNR2
SCHEMBL7549222 0.85 KDR (0.40) KDRFLT1FLT4ALPLCNR2
SCHEMBL7546645 0.85 FLT1 (0.40) KDRFLT1FLT4PDGFRBPDGFRA
SCHEMBL7551876 0.84 KDR (0.72) KDRFLT1FLT4CYP2A6PDGFRB
SCHEMBL7990118 0.84 KDR (0.39) KDRFLT1FLT4ALPLCNR2
SCHEMBL7991178 0.82 KDR (0.54) KDRFLT1FLT4CYP2A6PDGFRB
SCHEMBL7990971 0.81 KDR (0.70) KDRFLT1FLT4CYP2A6PDGFRB
SCHEMBL7547648 0.78 KDR (0.58) KDRFLT1FLT4CYP2A6
SCHEMBL7550794 0.78 KDR (0.56) KDRFLT1FLT4CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed