SCHEMBL7990615

SCHEMBL7990615

Cn1cc(C2=C(c3cn(C)c4cc(N5CCCC5)ccc34)C(=O)OC2=O)c2ccc(C#N)cc21

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.43
CREBBP Q92793 1/20 0.43
ALK Q9UM73 13/20 0.43
PGR P06401 1/20 0.39
GSK3B P49841 1/20 0.38
MEN1 O00255 1/20 0.37
ALDH1A1 P00352 1/20 0.37
MAPT P10636 1/20 0.37
ALOX15 P16050 1/20 0.37
KMT2A Q03164 1/20 0.37
HSD17B10 Q99714 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
USP14 P54578 1/20 0.36
KIT P10721 1/20 0.36
KDR P35968 1/20 0.36
SCN9A Q15858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7525540 0.87 ALK (0.49) BRD4CREBBPALKGSK3BMEN1
SCHEMBL7526149 0.81 GSK3B (0.53) BRD4CREBBPALKGSK3BKIT
SCHEMBL7976776 0.73 CDK4 (0.67) GSK3BMEN1MAPTKMT2A
SCHEMBL7987101 0.73 CDK4 (0.66) GSK3BMEN1MAPTKMT2A
SCHEMBL6952413 0.71 CCNE2 (0.71) GSK3B
SCHEMBL7524580 0.70 GSK3B (0.58) GSK3BMEN1MAPTKMT2A
SCHEMBL7529269 0.70 GSK3B (0.54) GSK3BMEN1MAPTKMT2A
SCHEMBL7990678 0.69 GSK3B (0.59) GSK3BKDR
SCHEMBL7497372 0.68 GSK3B (0.58) BRD4CREBBPGSK3B
SCHEMBL7523859 0.68 GSK3B (0.55) GSK3BMEN1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6281356-B1 ANTICANRCER AGENTS HOFFMANN-LA ROCHE INC. 2001-08-28 US disclosed