SCHEMBL7991002

SCHEMBL7991002

COc1cccc(-c2cncc(-c3cn(CCCN(C)C)c4cc(Cl)ccc34)c2)c1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDR P35968 4/20 0.53
GSK3B P49841 3/20 0.41
QPCT Q16769 1/20 0.41
ROCK1 Q13464 3/20 0.39
ROCK2 O75116 2/20 0.39
PRKCA P17252 2/20 0.39
PRKCB P05771 1/20 0.39
PRKCE Q02156 1/20 0.39
FLT3 P36888 1/20 0.39
PRKD1 Q15139 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
HTR6 P50406 2/20 0.38
FLT1 P17948 2/20 0.38
FLT4 P35916 2/20 0.38
BRD4 O60885 1/20 0.37
PRKACA P17612 1/20 0.36
PRKACG P22612 1/20 0.36
PRKACB P22694 1/20 0.36
ICMT O60725 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7546697 0.93 KDR (0.53) KDRGSK3BQPCTPRKCAPRKCB
SCHEMBL7976106 0.91 KDR (0.58) KDRPRKCAPRKCBPRKCEFLT3
SCHEMBL7988211 0.90 KDR (0.53) KDRGSK3BQPCTPRKCAPRKCB
SCHEMBL7550679 0.89 KDR (0.67) KDRGSK3BQPCTPRKCAPRKCB
SCHEMBL7550957 0.88 KDR (0.62) KDRPRKCAPRKCBPRKCEFLT3
SCHEMBL7993991 0.87 KDR (0.53) KDRGSK3BQPCTPRKCAPRKCB
SCHEMBL7987071 0.87 KDR (0.56) KDRGSK3BQPCTFLT3PRKD1
SCHEMBL7990452 0.85 KDR (0.58) KDRGSK3BPRKCAPRKCBPRKCE
SCHEMBL7548808 0.85 KDR (0.54) KDRGSK3BQPCTTDP1FLT1
SCHEMBL7552517 0.85 KDR (0.56) KDRGSK3BQPCTTDP1FLT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed