SCHEMBL7991229

SCHEMBL7991229

COc1ccc(COc2cc3c(cc2OC)C(C(=O)c2ccccc2)=NCC3)cc1

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.49
HPGD P15428 1/20 0.49
ATM Q13315 1/20 0.48
RAD52 P43351 1/20 0.48
GLA P06280 1/20 0.47
RCE1 Q9Y256 1/20 0.47
ALDH1A1 P00352 2/20 0.47
LMNA P02545 2/20 0.47
PTGER1 P34995 2/20 0.46
KMT2A Q03164 2/20 0.44
HSD17B10 Q99714 1/20 0.44
REV1 Q9UBZ9 1/20 0.42
MEN1 O00255 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
ACHE P22303 1/20 0.42
GRIN2C Q14957 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7977331 0.96 KDM4E (0.49) KDM4EHPGDATMRAD52GLA
SCHEMBL7988142 0.94 KDM4E (0.53) KDM4EHPGDATMRAD52GLA
SCHEMBL7991437 0.90 KDM4E (0.48) KDM4EHPGDATMRAD52GLA
SCHEMBL7991331 0.89 KDM4E (0.53) KDM4EHPGDATMRAD52GLA
SCHEMBL7992415 0.87 KDM4E (0.51) KDM4EHPGDATMRAD52GLA
SCHEMBL7994703 0.87 KDM4E (0.45) KDM4EHPGDATMRAD52GLA
SCHEMBL7987500 0.87 SMPD1 (0.53) KDM4EHPGDATMRAD52GLA
SCHEMBL7991324 0.84 KDM4E (0.56) KDM4EHPGDATMRAD52GLA
SCHEMBL7991327 0.83 KDM4E (0.52) KDM4EHPGDRAD52GLARCE1
SCHEMBL7988818 0.83 MAOB (0.48) NPC1RAB9AACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001055117-A1 NOVEL ISOQUINOLINE DERIVATIVES, PREPARATION METHOD AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM LES LABORATOIRES SERVIER (FR) 2001-08-02 WO disclosed