SCHEMBL7977331

SCHEMBL7977331

COc1ccc(C(=O)C2=NCCc3cc(OCc4ccccc4)c(OC)cc32)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.49
HPGD P15428 2/20 0.49
GLA P06280 1/20 0.49
RCE1 Q9Y256 1/20 0.49
ALDH1A1 P00352 2/20 0.47
LMNA P02545 1/20 0.47
ATM Q13315 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
RAD52 P43351 1/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
ACHE P22303 1/20 0.45
KMT2A Q03164 1/20 0.44
HSD17B10 Q99714 1/20 0.44
SMPD1 P17405 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC8 Q9BY41 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7991229 0.96 KDM4E (0.49) KDM4EHPGDGLARCE1ALDH1A1
SCHEMBL7988142 0.94 KDM4E (0.53) KDM4EHPGDGLARCE1ATM
SCHEMBL7991331 0.93 KDM4E (0.53) KDM4EHPGDGLARCE1ATM
SCHEMBL7987500 0.91 SMPD1 (0.53) KDM4EHPGDGLARCE1ATM
SCHEMBL7991437 0.90 KDM4E (0.48) KDM4EHPGDGLARCE1ATM
SCHEMBL7992415 0.87 KDM4E (0.51) KDM4EHPGDGLARCE1ATM
SCHEMBL7994703 0.87 KDM4E (0.45) KDM4EHPGDGLARCE1ATM
SCHEMBL7988818 0.87 MAOB (0.48) NPC1RAB9ASMN1; SMN2ACHE
SCHEMBL7991324 0.86 KDM4E (0.56) KDM4EHPGDGLARCE1ATM
SCHEMBL7989198 0.84 KDM4E (0.57) KDM4EHPGDGLARCE1RAD52

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001055117-A1 NOVEL ISOQUINOLINE DERIVATIVES, PREPARATION METHOD AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM LES LABORATOIRES SERVIER (FR) 2001-08-02 WO claimed
WO-2001055117-A1 NOVEL ISOQUINOLINE DERIVATIVES, PREPARATION METHOD AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM LES LABORATOIRES SERVIER (FR) 2001-08-02 WO disclosed