SCHEMBL7991720

SCHEMBL7991720

NC1(c2ccc(Br)cc2)CCC(=O)CC1

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 3/20 0.44
MEN1 O00255 1/20 0.39
CYP2C9 P11712 1/20 0.39
KMT2A Q03164 1/20 0.39
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
PIM1 P11309 1/20 0.34
PIM2 Q9P1W9 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL991567 0.83 CYP2A6 (0.42)
Hydrochloric Acid SCHEMBL5060581 0.81 KDM1A (0.40)
SCHEMBL10132207 0.80 MEN1 (0.39) HSD11B1MEN1CYP2C9KMT2AMAOA
SCHEMBL8005872 0.80 MAOB (0.39) HSD11B1MEN1CYP2C9KMT2AMAOA
SCHEMBL10241812 0.79 MAOA (0.36) HSD11B1MEN1KMT2AMAOAMAOB
SCHEMBL614021 0.79 MEN1 (0.63) MEN1CYP2C9KMT2A
SCHEMBL9966307 0.79 AKT1 (0.41)
SCHEMBL255382 0.79 AKT2 (0.44)
Hydrochloric Acid SCHEMBL5767667 0.78 MAOB (0.38) HSD11B1MEN1CYP2C9KMT2AMAOA
Hydrochloric Acid SCHEMBL5383464 0.78 MEN1 (0.61) MEN1CYP2C9KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009156100-A1 SUBSTITUTED ISOQUINOLINES AND ISOQUINOLINONES AS RHO KINASE INHIBITORS SANOFI-AVENTIS (FR) 2009-12-30 WO disclosed