SCHEMBL7992108

SCHEMBL7992108

N=C(N)NC(=O)c1ccc(C2CCN(C(=O)[C@@H](N)CCC=O)CC2)c(C(F)(F)F)c1

nearest known ligand 0.49

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SLC9A1 P19634 19/20 0.49
CYP2C9 P11712 10/20 0.49
CYP3A4 P08684 6/20 0.49
CYP2C19 P33261 8/20 0.45
ADRA1D P25100 2/20 0.45
SLC6A3 Q01959 2/20 0.45
HTR2A P28223 1/20 0.45
SLC9A2 Q9UBY0 1/20 0.45
CYP2D6 P10635 3/20 0.44
KCNH2 Q12809 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7980132 0.88 SLC9A1 (0.53) SLC9A1CYP2C9CYP3A4CYP2C19ADRA1D
SCHEMBL1764258 0.88 SLC9A1 (0.53) SLC9A1CYP2C9CYP3A4CYP2C19ADRA1D
SCHEMBL1763714 0.88 SLC9A1 (0.52) SLC9A1CYP2C9CYP3A4CYP2C19ADRA1D
SCHEMBL1764116 0.87 SLC9A1 (0.51) SLC9A1CYP2C9CYP3A4CYP2C19ADRA1D
SCHEMBL1763946 0.87 SLC9A1 (0.52) SLC9A1CYP2C9CYP3A4CYP2C19ADRA1D
SCHEMBL1763717 0.87 SLC9A1 (0.52) SLC9A1CYP2C9CYP3A4CYP2C19ADRA1D
SCHEMBL1763654 0.86 SLC9A1 (0.50) SLC9A1CYP2C9CYP3A4CYP2C19ADRA1D
SCHEMBL1763657 0.86 SLC9A1 (0.50) SLC9A1CYP2C9CYP3A4CYP2C19ADRA1D
SCHEMBL1763483 0.86 SLC9A1 (0.55) SLC9A1CYP2C9CYP3A4CYP2C19ADRA1D
SCHEMBL1763570 0.85 SLC9A1 (0.52) SLC9A1CYP2C9CYP3A4CYP2C19ADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010005783-A1 PYRROLIDINYL AND PIPERIDINYL COMPOUNDS USEFUL AS NHE-1 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-01-14 WO disclosed