SCHEMBL7992800

SCHEMBL7992800

O=C(Cl)CN1CN(c2ccccc2)C2(CCN(Cc3cccc4ccccc34)CC2)C1=O

nearest known ligand 0.78

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 9/20 0.78
MEN1 O00255 1/20 0.54
CYP3A4 P08684 1/20 0.54
CYP2D6 P10635 1/20 0.54
CYP2C9 P11712 1/20 0.54
KMT2A Q03164 1/20 0.54
DRD2 P14416 6/20 0.54
DRD3 P35462 6/20 0.54
DRD4 P21917 5/20 0.54
OPRM1 P35372 8/20 0.53
OPRD1 P41143 8/20 0.53
OPRK1 P41145 8/20 0.53
BDKRB2 P30411 1/20 0.52
DDR1 Q08345 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7754117 0.92 OPRL1 (0.81) OPRL1MEN1CYP3A4CYP2D6CYP2C9
SCHEMBL29766745 0.88 OPRL1 (1.00) OPRL1MEN1CYP3A4CYP2D6CYP2C9
SCHEMBL7757872 0.88 OPRL1 (1.00) OPRL1MEN1CYP3A4CYP2D6CYP2C9
SCHEMBL7992795 0.87 OPRL1 (0.76) OPRL1MEN1CYP3A4CYP2D6CYP2C9
SCHEMBL7754142 0.86 OPRL1 (0.74) OPRL1MEN1CYP3A4CYP2D6CYP2C9
SCHEMBL7754138 0.85 OPRL1 (0.72) OPRL1MEN1CYP3A4CYP2D6CYP2C9
SCHEMBL7754144 0.85 OPRL1 (0.72) OPRL1MEN1CYP3A4CYP2D6CYP2C9
SCHEMBL5108205 0.85 OPRL1 (0.72) OPRL1MEN1CYP3A4CYP2D6CYP2C9
SCHEMBL7999928 0.84 OPRL1 (0.67) OPRL1DRD2DRD3DRD4OPRM1
Hydrochloric Acid SCHEMBL7758893 0.84 OPRL1 (0.71) OPRL1MEN1CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001036418-A1 NOVEL TRIAZASPIRODECANONES WITH HIGH AFFINITY FOR OPIOID RECEPTOR SUBTYPES NOVO NORDISK A/S (DK) 2001-05-25 WO disclosed