SCHEMBL7994425

SCHEMBL7994425

CC(C)(C)C#Cc1ccc(C(CCO)c2c[nH]cn2)cc1

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.37
HAO1 Q9UJM8 1/20 0.33
EGLN1 Q9GZT9 1/20 0.31
FNTA P49354 1/20 0.30
FNTB P49356 1/20 0.30
PGGT1B P53609 1/20 0.30
CYP2D6 P10635 1/20 0.30
HRH4 Q9H3N8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4387548 0.86 HRH3 (0.36) HRH3HAO1FNTAFNTBPGGT1B
SCHEMBL4387545 0.72 HRH3 (0.36) HRH3HAO1
SCHEMBL4388946 0.66
SCHEMBL2105057 0.65 CHRM2 (0.41) CYP2D6
SCHEMBL9090439 0.64 CYP19A1 (0.55)
SCHEMBL7991000 0.64 HRH3 (0.39) HRH3HAO1CYP2D6
SCHEMBL4954449 0.63 HRH3 (0.47) HRH3HAO1EGLN1CYP2D6HRH4
SCHEMBL2104158 0.63 CHRM2 (0.41) HRH3CYP2D6
SCHEMBL9090407 0.62 CYP19A1 (0.62)
SCHEMBL6588101 0.62 RIPK1 (0.38) CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6248765-B1 ANTIINFLAMMATORY AGENTS; HYPOTENSIVE AGENTS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICAL (FR) 2001-06-19 US claimed