SCHEMBL7994756

SCHEMBL7994756

N=C(N)NC(=O)c1ccc(C2CCN(C(=O)c3ccc(N)cc3)CC2)c(C(F)(F)F)c1

nearest known ligand 0.62

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SLC9A1 P19634 20/20 0.62
CYP2C9 P11712 8/20 0.59
CYP2C19 P33261 5/20 0.59
CYP3A4 P08684 5/20 0.59
CYP2D6 P10635 2/20 0.59
KCNH2 Q12809 1/20 0.55
ADRA1D P25100 1/20 0.51
HTR2A P28223 1/20 0.51
SLC6A3 Q01959 1/20 0.51
SLC9A2 Q9UBY0 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1763892 0.93 SLC9A1 (0.68) SLC9A1CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL1763080 0.93 SLC9A1 (0.68) SLC9A1CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL1763943 0.92 SLC9A1 (0.69) SLC9A1CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL1763920 0.92 SLC9A1 (0.69) SLC9A1CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL1763620 0.92 SLC9A1 (0.62) SLC9A1CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL1763519 0.92 SLC9A1 (0.69) SLC9A1CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL8000352 0.91 SLC9A1 (0.58) SLC9A1CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL1763600 0.91 SLC9A1 (0.75) SLC9A1CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL1763899 0.91 SLC9A1 (0.69) SLC9A1CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL1763606 0.91 SLC9A1 (0.69) SLC9A1CYP2C9CYP2C19CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010005783-A1 PYRROLIDINYL AND PIPERIDINYL COMPOUNDS USEFUL AS NHE-1 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-01-14 WO disclosed