SCHEMBL7994898

SCHEMBL7994898

N=C(N)NC(=O)c1ccc(C2CCN(C(=O)c3ccc(-c4cccc(O)c4)nc3)CC2)c(C(F)(F)F)c1

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SLC9A1 P19634 20/20 0.50
CYP2C9 P11712 10/20 0.50
CYP2C19 P33261 7/20 0.48
CYP2D6 P10635 3/20 0.47
CYP3A4 P08684 5/20 0.47
KCNH2 Q12809 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1763479 0.89 SLC9A1 (0.48) SLC9A1CYP2C9CYP2C19CYP2D6CYP3A4
SCHEMBL1764067 0.89 SLC9A1 (0.53) SLC9A1CYP2C9CYP2C19CYP2D6CYP3A4
SCHEMBL1763547 0.87 SLC9A1 (0.55) SLC9A1CYP2C9CYP2C19CYP2D6CYP3A4
SCHEMBL1763255 0.86 SLC9A1 (0.56) SLC9A1CYP2C9CYP2C19CYP2D6CYP3A4
SCHEMBL7993065 0.85 SLC9A1 (0.55) SLC9A1CYP2C9CYP2C19CYP2D6CYP3A4
SCHEMBL1763647 0.85 SLC9A1 (0.59) SLC9A1CYP2C9CYP2C19CYP2D6CYP3A4
SCHEMBL1763920 0.84 SLC9A1 (0.69) SLC9A1CYP2C9CYP2C19CYP2D6CYP3A4
SCHEMBL1763826 0.83 SLC9A1 (0.70) SLC9A1CYP2C9CYP2C19CYP2D6CYP3A4
SCHEMBL8000752 0.82 SLC9A1 (0.54) SLC9A1CYP2C9CYP2C19CYP2D6CYP3A4
SCHEMBL1763931 0.82 SLC9A1 (0.72) SLC9A1CYP2C9CYP2C19CYP2D6CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010005783-A1 PYRROLIDINYL AND PIPERIDINYL COMPOUNDS USEFUL AS NHE-1 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-01-14 WO disclosed