SCHEMBL7995059

SCHEMBL7995059

COc1ccccc1-c1cc(C)ccn1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 1/20 0.56
ADRA1A P35348 1/20 0.56
ADRA1B P35368 1/20 0.56
CCR1 P32246 1/20 0.53
CCR5 P51681 1/20 0.53
CCR8 P51685 1/20 0.53
CYP1A2 P05177 7/20 0.51
CYP2C19 P33261 7/20 0.51
ALDH1A1 P00352 7/20 0.51
CYP2D6 P10635 6/20 0.51
CLK4 Q9HAZ1 6/20 0.51
CYP3A4 P08684 5/20 0.51
LMNA P02545 5/20 0.51
TSHR P16473 5/20 0.51
HSD17B10 Q99714 5/20 0.51
MAPK1 P28482 4/20 0.50
HSP90AA1 P07900 1/20 0.50
KDM1A O60341 1/20 0.49
HDAC1 Q13547 1/20 0.49
HDAC6 Q9UBN7 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28452211 0.81 HSP90AA1 (0.53) CYP1A2CYP2C19ALDH1A1CYP2D6CLK4
SCHEMBL28987610 0.79 KDM1A (0.46) CYP1A2CYP2C19ALDH1A1CYP2D6CLK4
SCHEMBL987521 0.78 CCR1 (0.61) ADRA1DADRA1AADRA1BCCR1CCR5
SCHEMBL29496935 0.78 SMN1; SMN2 (0.62) ADRA1DADRA1AADRA1BCCR1CCR5
SCHEMBL2039527 0.78 SMN1; SMN2 (0.62) ADRA1DADRA1AADRA1BCCR1CCR5
SCHEMBL15344911 0.78 CCR1 (0.52) ADRA1DADRA1AADRA1BCCR1CCR5
SCHEMBL4765389 0.78 FYN (0.51) CYP1A2CYP2C19ALDH1A1CYP2D6CLK4
SCHEMBL4128874 0.78 CYP1A2 (0.48) CYP1A2CYP2C19ALDH1A1CYP2D6CLK4
SCHEMBL13801591 0.77 CCR1 (0.59) ADRA1DADRA1AADRA1BCCR1CCR5
SCHEMBL15476086 0.77 CCR1 (0.59) ADRA1DADRA1AADRA1BCCR1CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010005783-A1 PYRROLIDINYL AND PIPERIDINYL COMPOUNDS USEFUL AS NHE-1 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-01-14 WO disclosed