SCHEMBL7998430

SCHEMBL7998430

Nc1ccc2c(c1)C[C@@H](NC(=O)OCc1ccccc1)C2

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.58
ALDH1A1 P00352 2/20 0.57
GAA P10253 1/20 0.57
CA1 P00915 2/20 0.56
CA2 P00918 2/20 0.56
ACHE P22303 2/20 0.56
CTSL P07711 1/20 0.50
CTSB P07858 1/20 0.50
CTSK P43235 1/20 0.50
EPHX1 P07099 1/20 0.49
DPP4 P27487 3/20 0.46
DPP7 Q9UHL4 3/20 0.46
KCNH2 Q12809 1/20 0.46
HDAC8 Q9BY41 1/20 0.45
CPB1 P15086 1/20 0.45
PSEN1 P49768 1/20 0.44
PSEN2 P49810 1/20 0.44
APH1B Q8WW43 1/20 0.44
NCSTN Q92542 1/20 0.44
APH1A Q96BI3 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL170233 0.87 ALDH1A1 (0.65) TSHRALDH1A1GAACA1CA2
SCHEMBL7902024 0.85 CA1 (0.56) TSHRALDH1A1GAACA1CA2
SCHEMBL7967064 0.85 CA1 (0.56) TSHRALDH1A1GAACA1CA2
SCHEMBL614655 0.85 CA1 (0.56) TSHRALDH1A1GAACA1CA2
SCHEMBL12633938 0.85 CA1 (0.56) TSHRALDH1A1GAACA1CA2
SCHEMBL12633934 0.85 CA1 (0.56) TSHRALDH1A1GAACA1CA2
SCHEMBL614654 0.85 CA1 (0.56) TSHRALDH1A1GAACA1CA2
SCHEMBL12633937 0.85 CA1 (0.56) TSHRALDH1A1GAACA1CA2
SCHEMBL7973199 0.85 CA1 (0.56) TSHRALDH1A1GAACA1CA2
SCHEMBL7898004 0.84 CA1 (0.55) TSHRALDH1A1GAACA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009105026-A1 COMPOUND (R) -N*6*-ETHYL-6, 7-DIHYDRO-5H-INDENO (5, 6- D) THIAZOLE-2, 6-DIAMINE AND THE USE AS ANTIPSYCHOTICS ASTRAZENECA AB (SE) 2009-08-27 WO disclosed