SCHEMBL7998657

SCHEMBL7998657

Cn1cnc(NCc2ccccc2)c2ncnc1-2

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 5/20 0.59
KDM4E B2RXH2 2/20 0.54
TMIGD3 P0DMS9 1/20 0.48
ADORA2A P29274 1/20 0.48
ADORA1 P30542 1/20 0.48
HTT P42858 2/20 0.48
CCNB2 O95067 2/20 0.46
CCNB1 P14635 2/20 0.46
CDK2 P24941 2/20 0.46
CCNB3 Q8WWL7 2/20 0.46
EGFR P00533 2/20 0.46
RAB9A P51151 2/20 0.46
GALR3 O60755 2/20 0.46
NR2F2 P24468 2/20 0.46
KMT2A Q03164 2/20 0.45
MAPK1 P28482 3/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
CYP1A2 P05177 2/20 0.44
CYP2D6 P10635 2/20 0.44
TSHR P16473 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20880133 0.80 KDM4E (0.61) CDK1KDM4ETMIGD3ADORA2AADORA1
SCHEMBL21121655 0.75 SMN1; SMN2 (0.55) CDK1KDM4ETMIGD3ADORA2AADORA1
SCHEMBL4382069 0.74 CDK1 (1.00) CDK1KDM4ETMIGD3ADORA2AADORA1
SCHEMBL8011473 0.74 CDK1 (0.63) CDK1KDM4ETMIGD3ADORA2AADORA1
SCHEMBL1387903 0.72 ALDH1A1 (0.43) CDK1TMIGD3ADORA2AADORA1HTT
SCHEMBL7382606 0.72 TMIGD3 (0.49) KDM4ETMIGD3ADORA2AADORA1EGFR
SCHEMBL9567831 0.70 AURKA (0.40) CDK1KDM4EHTTCCNB2CCNB1
SCHEMBL24667246 0.69 CDK1 (0.63) CDK1KDM4ETMIGD3ADORA2AADORA1
SCHEMBL1388236 0.69 PDE4A (0.52) ADORA2AHTTSMN1; SMN2ALDH1A1
SCHEMBL28829351 0.69 FLT1 (0.60) CDK1KDM4ECCNB2CCNB1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000033657-A1 METHOD TO IDENTIFY REGULATORS OF CDK ACTIVITY CROPDESIGN N.V. (BE) 2000-06-15 WO claimed
WO-2000033657-A1 METHOD TO IDENTIFY REGULATORS OF CDK ACTIVITY CROPDESIGN N.V. (BE) 2000-06-15 WO disclosed