SCHEMBL7999897

SCHEMBL7999897

CN1C(=O)C2CNCC2(c2cccc(Br)c2)N/C1=N/C(=O)OC(C)(C)C

nearest known ligand 0.35

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
RORC P51449 2/20 0.35
GRM5 P41594 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12649761 0.89 GRM5 (0.33) GRM5
SCHEMBL8002607 0.89 RORC (0.36) RORC
SCHEMBL8247691 0.87 RORC (0.36) RORCGRM5
SCHEMBL12649654 0.87 GRM5 (0.36) GRM5
SCHEMBL12947092 0.84 BACE1 (0.39) GRM5
SCHEMBL12916796 0.84 BACE1 (0.39) GRM5
SCHEMBL12649758 0.80 SCN9A (0.34)
SCHEMBL12649715 0.80
SCHEMBL12649778 0.79
SCHEMBL12649759 0.79

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2288613-B1 PHENYL-SUBSTITUTED 2-IMINO-3-METHYL PYRROLO PYRIMIDINONE COMPOUNDS AS BACE-1 INHIBITORS, COMPOSITIONS, AND THEIR USE MERCK SHARP & DOHME (US) 2016-07-13 EP disclosed
WO-2009131975-A1 PHENYL-SUBSTITUTED 2-IMINO-3-METHYL PYRROLO PYRIMIDINONE COMPOUNDS AS BACE-1 INHIBITORS, COMPOSITIONS, AND THEIR USE SCHERING CORPORATION (US) 2009-10-29 WO disclosed