SCHEMBL8000384

SCHEMBL8000384

COc1ccc(C[C@@H](N)C(=O)O)cc1Br

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 1/20 0.56
CD274 Q9NZQ7 1/20 0.56
LDHA P00338 1/20 0.55
TPH1 P17752 8/20 0.54
SLC7A5 Q01650 4/20 0.53
KDM4E B2RXH2 2/20 0.53
TDP1 Q9NUW8 2/20 0.53
USP2 O75604 1/20 0.53
EGFR P00533 1/20 0.53
LCK P06239 1/20 0.53
FYN P06241 1/20 0.53
ADORA3 P0DMS8 1/20 0.53
ALOX15 P16050 1/20 0.53
PTGS1 P23219 1/20 0.53
HTR2A P28223 1/20 0.53
PTGS2 P35354 1/20 0.53
RECQL P46063 1/20 0.53
HIF1A Q16665 1/20 0.53
HSD17B10 Q99714 1/20 0.53
NR1I2 O75469 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15760890 1.00 PDCD1 (0.56) PDCD1CD274LDHATPH1SLC7A5
SCHEMBL6339536 1.00 PDCD1 (0.56) PDCD1CD274LDHATPH1SLC7A5
SCHEMBL8009937 0.86 LDHA (0.73) LDHATPH1SLC7A5KDM4ETDP1
SCHEMBL31242504 0.86 LDHA (0.73) LDHATPH1SLC7A5KDM4ETDP1
SCHEMBL30013904 0.86 LDHA (0.73) LDHATPH1SLC7A5KDM4ETDP1
SCHEMBL159001 0.86 LDHA (0.73) LDHATPH1SLC7A5KDM4ETDP1
SCHEMBL159000 0.86 LDHA (0.73) LDHATPH1SLC7A5KDM4ETDP1
SCHEMBL29637606 0.86 LDHA (0.73) LDHATPH1SLC7A5KDM4ETDP1
Hydrochloric Acid SCHEMBL10464213 0.85 LDHA (0.71) LDHATPH1SLC7A5KDM4ETDP1
Hydrochloric Acid SCHEMBL3207583 0.85 LDHA (0.71) LDHATPH1SLC7A5KDM4ETDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0850316-A4 CRYPTOPHYCINS FROM ABERRANT BIOSYNTHESIS UNIV HAWAII (US) 2000-08-23 EP disclosed
EP-0850316-A1 CRYPTOPHYCINS FROM ABERRANT BIOSYNTHESIS UNIVERSITY OF HAWAII (US) 1998-07-01 EP disclosed
WO-1997008334-A1 CRYPTOPHYCINS FROM ABERRANT BIOSYNTHESIS UNIVERSITY OF HAWAII (US) 1997-03-06 WO disclosed