SCHEMBL8000516

SCHEMBL8000516

CC(=O)NCCc1ccc(/C(Nc2ccc(-c3c[nH]c(N4CCCCC4)n3)cc2)=C2/C(=O)Nc3ccc([N+](=O)[O-])cc32)cc1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
CNR1 P21554 2/20 0.35
AKT2 P31751 4/20 0.34
PDPK1 O15530 3/20 0.34
MEN1 O00255 2/20 0.34
NQO2 P16083 1/20 0.34
CA12 O43570 2/20 0.33
CA1 P00915 2/20 0.33
CA2 P00918 2/20 0.33
CA9 Q16790 2/20 0.33
EGFR P00533 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8000521 1.00 KMT2A (0.35) KMT2ANPC1RAB9ACNR1AKT2
SCHEMBL8012266 0.96 KMT2A (0.36) KMT2ANPC1RAB9ACNR1AKT2
SCHEMBL8012262 0.96 KMT2A (0.36) KMT2ANPC1RAB9ACNR1AKT2
SCHEMBL8017092 0.90 CNR1 (0.36) KMT2ANPC1RAB9ACNR1AKT2
SCHEMBL8017088 0.90 CNR1 (0.36) KMT2ANPC1RAB9ACNR1AKT2
SCHEMBL8009531 0.90 NQO2 (0.38) KMT2ANPC1RAB9ACNR1AKT2
SCHEMBL8009527 0.90 NQO2 (0.38) KMT2ANPC1RAB9ACNR1AKT2
SCHEMBL8009854 0.90 HRH3 (0.37) KMT2ACNR1AKT2PDPK1MEN1
SCHEMBL8009849 0.90 HRH3 (0.37) KMT2ACNR1AKT2PDPK1MEN1
SCHEMBL8009901 0.89 CNR1 (0.35) KMT2ACNR1AKT2PDPK1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6043254-A ANTIPROLIFERATIVE AGENT; ENZYME INHIBITOR BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-03-28 US disclosed