SCHEMBL8009901

SCHEMBL8009901

NCCCc1ccc(C(Nc2ccc(-c3c[nH]c(N4CCCCC4)n3)cc2)=C2C(=O)Nc3ccc([N+](=O)[O-])cc32)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.35
CA12 O43570 2/20 0.34
CA1 P00915 2/20 0.34
CA2 P00918 2/20 0.34
CA9 Q16790 2/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
EGFR P00533 1/20 0.34
CASP3 P42574 3/20 0.32
CAPN9 O14815 1/20 0.32
ALDH1A1 P00352 4/20 0.31
MAPT P10636 2/20 0.31
GAA P10253 2/20 0.31
PDPK1 O15530 1/20 0.31
AKT2 P31751 1/20 0.31
POLB P06746 1/20 0.31
MPI P34949 1/20 0.31
BLM P54132 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
CYP3A4 P08684 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8009896 1.00 CNR1 (0.35) CNR1CA12CA1CA2CA9
SCHEMBL8017092 0.96 CNR1 (0.36) CNR1CA12CA1CA2CA9
SCHEMBL8017088 0.96 CNR1 (0.36) CNR1CA12CA1CA2CA9
SCHEMBL8009405 0.93 MEN1 (0.36) CNR1CA12CA1CA2CA9
SCHEMBL8009411 0.93 MEN1 (0.36) CNR1CA12CA1CA2CA9
SCHEMBL8009854 0.91 HRH3 (0.37) CNR1CA12CA1CA2CA9
SCHEMBL8009849 0.91 HRH3 (0.37) CNR1CA12CA1CA2CA9
SCHEMBL8012266 0.90 KMT2A (0.36) CNR1CA12CA1CA2CA9
SCHEMBL8012262 0.90 KMT2A (0.36) CNR1CA12CA1CA2CA9
SCHEMBL8000714 0.90 CASP1 (0.40) CNR1CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6043254-A ANTIPROLIFERATIVE AGENT; ENZYME INHIBITOR BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-03-28 US disclosed