SCHEMBL8000714

SCHEMBL8000714

O=C1Nc2ccc([N+](=O)[O-])cc2/C1=C(/Nc1ccc(-c2c[nH]c(N3CCCC3)n2)cc1)c1ccc(CN2CCCCC2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 1/20 0.40
CASP4 P49662 1/20 0.40
CASP5 P51878 1/20 0.40
ALDH1A1 P00352 3/20 0.36
MAPT P10636 2/20 0.36
CNR1 P21554 1/20 0.36
EGFR P00533 1/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34
CDK4 P11802 1/20 0.34
CCND1 P24385 1/20 0.34
ROCK2 O75116 1/20 0.34
CCR2 P41597 1/20 0.34
ROCK1 Q13464 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
MAP3K7 O43318 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8000723 1.00 CASP1 (0.40) CASP1CASP4CASP5ALDH1A1MAPT
SCHEMBL8012613 0.99 CASP1 (0.40) CASP1CASP4CASP5ALDH1A1MAPT
SCHEMBL8012609 0.99 CASP1 (0.40) CASP1CASP4CASP5ALDH1A1MAPT
SCHEMBL8009854 0.93 HRH3 (0.37) ALDH1A1CNR1EGFRMEN1KMT2A
SCHEMBL8009849 0.93 HRH3 (0.37) ALDH1A1CNR1EGFRMEN1KMT2A
SCHEMBL8010035 0.93 CASP1 (0.39) CASP1CASP4CASP5ALDH1A1MAPT
SCHEMBL8010033 0.93 CASP1 (0.39) CASP1CASP4CASP5ALDH1A1MAPT
SCHEMBL8009241 0.93 IRAK4 (0.35) CASP1CASP4CASP5ALDH1A1MAPT
SCHEMBL8009239 0.93 IRAK4 (0.35) CASP1CASP4CASP5ALDH1A1MAPT
SCHEMBL8001515 0.92 CASP1 (0.39) CASP1CASP4CASP5ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6043254-A ANTIPROLIFERATIVE AGENT; ENZYME INHIBITOR BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-03-28 US disclosed