SCHEMBL8001497

SCHEMBL8001497

O=C(O)CCCc1c(Cc2ccccc2)[nH]c2ccccc12

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 3/20 0.63
MTNR1B P49286 3/20 0.63
CYP1A2 P05177 2/20 0.63
CYP3A4 P08684 2/20 0.63
HPGD P15428 2/20 0.63
TSHR P16473 2/20 0.63
CYP2C19 P33261 2/20 0.63
TDP1 Q9NUW8 2/20 0.63
MEN1 O00255 2/20 0.63
KMT2A Q03164 2/20 0.63
CYP2C9 P11712 1/20 0.63
EGFR P00533 3/20 0.63
ALDH1A1 P00352 4/20 0.62
MAPT P10636 2/20 0.62
CYP2D6 P10635 1/20 0.62
ALOX15 P16050 1/20 0.62
MC4R P32245 4/20 0.57
MC5R P33032 4/20 0.57
MC3R P41968 4/20 0.57
KDM4E B2RXH2 4/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2944735 0.92 MTNR1A (0.66) MTNR1AMTNR1BCYP1A2CYP3A4HPGD
SCHEMBL2087168 0.82 HPGD (0.61) MTNR1AMTNR1BCYP1A2CYP3A4HPGD
SCHEMBL9368557 0.81 FFAR1 (0.47) MTNR1AMTNR1BCYP1A2CYP3A4HPGD
SCHEMBL30547373 0.80 EGFR (0.62) MTNR1AMTNR1BCYP1A2CYP3A4HPGD
SCHEMBL9153503 0.80 KDM4E (0.69) CYP3A4TSHRTDP1EGFRALDH1A1
SCHEMBL31034424 0.78 HPGD (0.58) MTNR1AMTNR1BCYP1A2CYP3A4HPGD
SCHEMBL25276059 0.78 EGFR (0.68) MEN1KMT2AEGFRALDH1A1MAPT
SCHEMBL28472093 0.78 OXER1 (0.61) HPGDMEN1KMT2AEGFRALDH1A1
SCHEMBL28190374 0.78 EGFR (0.68) MEN1KMT2AEGFRALDH1A1MAPT
SCHEMBL3276610 0.78 KDM4E (0.83) EGFRALDH1A1KDM4EGPR17

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000029022-A1 COX-2 INHIBITORS IN COMBINATION WITH CENTRALLY ACTING ANALGESICS ALGOS PHARMACEUTICAL CORPORATION (US) 2000-05-25 WO claimed