SCHEMBL8002483

SCHEMBL8002483

FC(F)(F)c1ccc(-c2ccc(-c3cccs3)cc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 6/20 0.56
LTA4H P09960 1/20 0.52
KCNH2 Q12809 1/20 0.50
TP53 P04637 1/20 0.48
CYP17A1 P05093 1/20 0.46
CYP11B1 P15538 1/20 0.46
CYP11B2 P19099 1/20 0.46
AGXT P21549 1/20 0.45
PDK2 Q15119 1/20 0.44
DRD4 P21917 1/20 0.43
HTR2A P28223 1/20 0.43
ERN1 O75460 2/20 0.43
CYP2E1 P05181 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2A6 P11509 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2B6 P20813 1/20 0.42
LPL P06858 1/20 0.42
LIPG Q9Y5X9 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL154628 0.98 LTA4H (0.53) KIF11LTA4HKCNH2TP53CYP17A1
SCHEMBL10472463 0.85 ERBB2 (0.46) KIF11LTA4HKCNH2TP53
SCHEMBL7455134 0.84 LTA4H (0.67) LTA4HKCNH2CYP17A1CYP11B1CYP11B2
SCHEMBL154838 0.84 CNR2 (0.50) LTA4HKCNH2TP53ERN1CYP2E1
SCHEMBL16546585 0.84 LTA4H (0.48) LTA4HKCNH2TP53CYP17A1CYP11B1
SCHEMBL338810 0.82 LTA4H (0.70) LTA4HKCNH2CYP17A1CYP11B1CYP11B2
SCHEMBL935372 0.82 ERN1 (0.49) LTA4HKCNH2TP53PDK2ERN1
SCHEMBL20368756 0.81 LTA4H (0.46) LTA4HKCNH2TP53CYP17A1CYP11B1
SCHEMBL28222643 0.80 ERN1 (0.51) KIF11LTA4HKCNH2CYP17A1CYP11B1
SCHEMBL1623633 0.79 LTA4H (0.52) KIF11LTA4HKCNH2TP53CYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6294573-B1 FOR THERAPY RHEUMATOID ARTHRITIS, OSTEOARTHRITIS, OSTEOPENIAS SUCH AS OSTEOPOROSIS, PERIODONTITIS, GINGIVITIS, CORNEAL, EPIDERMAL OR GASTRIC ULCERATION, AND TUMOR GROWTH AND METASTASIS OR INVASION ABBOTT LABORATORIES 2001-09-25 US disclosed