SCHEMBL8002912

SCHEMBL8002912

COc1ccc2c(N)cc(-c3cc(C(C)C)on3)nc2c1Cl

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.38
MEN1 O00255 1/20 0.38
CYP1A2 P05177 1/20 0.38
MAPK1 P28482 1/20 0.38
CYP2C19 P33261 1/20 0.38
KMT2A Q03164 1/20 0.38
SMN1; SMN2 Q16637 3/20 0.35
HPGD P15428 2/20 0.34
KDM4E B2RXH2 2/20 0.34
MAPT P10636 1/20 0.34
STAT3 P40763 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
G6PD P11413 1/20 0.34
CYP19A1 P11511 2/20 0.33
CYP11B1 P15538 2/20 0.33
CYP11B2 P19099 2/20 0.33
S1PR1 P21453 1/20 0.32
SLC2A1 P11166 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10271656 0.89 ALDH1A1 (0.40) ALDH1A1MEN1CYP1A2MAPK1CYP2C19
SCHEMBL10220691 0.88 ALDH1A1 (0.38) ALDH1A1MEN1CYP1A2MAPK1CYP2C19
SCHEMBL8007996 0.87 ALDH1A1 (0.36) ALDH1A1MEN1CYP1A2MAPK1CYP2C19
SCHEMBL314362 0.86 ALDH1A1 (0.40) ALDH1A1MEN1CYP1A2MAPK1CYP2C19
SCHEMBL7995957 0.86 ALDH1A1 (0.36) ALDH1A1MEN1CYP1A2MAPK1CYP2C19
SCHEMBL15216094 0.86 SLC2A1 (0.37) ALDH1A1MEN1CYP1A2MAPK1CYP2C19
SCHEMBL16579241 0.83 ALDH1A1 (0.37) ALDH1A1MEN1CYP1A2MAPK1CYP2C19
SCHEMBL8008865 0.78 ALDH1A1 (0.40) ALDH1A1MEN1KMT2ASMN1; SMN2KDM4E
SCHEMBL7995961 0.78 SLC2A1 (0.43) ALDH1A1MEN1CYP1A2MAPK1CYP2C19
SCHEMBL577561 0.77 ALDH1A1 (0.38) ALDH1A1MEN1CYP1A2MAPK1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009099596-A2 MACROCYCLIC SERINE PROTEASE INHIBITORS IDENIX PHARAMACEUTICALS, INC. (US) 2009-08-13 WO disclosed