SCHEMBL8003063

SCHEMBL8003063

CN(C)C[C@@H]1CCc2ccccc2C1=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
METAP1 P53582 4/20 0.71
CYP19A1 P11511 2/20 0.55
THRA P10827 1/20 0.53
THRB P10828 1/20 0.53
HTR1A P08908 1/20 0.50
SIGMAR1 Q99720 1/20 0.50
ACHE P22303 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2125675 1.00 METAP1 (0.71) METAP1CYP19A1THRATHRBHTR1A
Hydrochloric Acid SCHEMBL2125507 0.98 METAP1 (0.72) METAP1CYP19A1THRATHRB
SCHEMBL3822940 0.91 METAP1 (0.68) METAP1CYP19A1SIGMAR1ACHE
Hydrochloric Acid SCHEMBL2126669 0.89 METAP1 (0.68) METAP1SIGMAR1ACHE
SCHEMBL8489825 0.84 CYP19A1 (0.57) METAP1CYP19A1HTR1ASIGMAR1ACHE
SCHEMBL11635436 0.84 CYP19A1 (0.52) METAP1CYP19A1HTR1ASIGMAR1ACHE
Hydrochloric Acid SCHEMBL7706188 0.84 CYP19A1 (0.56) METAP1CYP19A1HTR1ASIGMAR1ACHE
SCHEMBL6630621 0.84 METAP1 (0.51) METAP1CYP19A1HTR1ASIGMAR1ACHE
SCHEMBL2175676 0.83 METAP1 (1.00) METAP1CYP19A1ACHE
SCHEMBL6630617 0.83 METAP1 (0.50) METAP1CYP19A1HTR1ASIGMAR1ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6022895-A Substituted amino compounds and their use as substances having an analgesic effect GRUENENTHAL GMBH (DE) 2000-02-08 US disclosed